IP Library Granted Patent US 10,919,962
Granted Patent B2
US 10,919,962 · App. 16/192,537 · Granted Feb 16, 2021

Method of reducing tumor growth with IL-1beta neutralizing human monoclonal antibodies

Inventors: Cheng-I Wang (Singapore, SG); Angeline Goh (Singapore, SG); Siok Ping Yeo (Singapore, SG); Alessandra Rosa Mortellaro (Singapore, SG); Subhra Kumar Biswas (Singapore, SG); Florent Ginhoux (Singapore, SG); Pingyu Zhong (Singapore, SG)
Assignee: Agency for Science, Technology and Research
C07K16/245A61K39/3955A61K2039/505C07K2317/10C07K2317/55C07K2317/56C07K2317/565C07K2317/73C07K2317/76C07K2317/92
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Quick Facts
Patent No.
US 10,919,962
App. No.
16/192,537
Granted
Feb 16, 2021
Kind
B2
Abstract

The present invention is directed to antigen binding proteins and in particular to IL-1β antigen binding proteins. The present invention further provides compositions comprising the antigen binding proteins, use of the antigen binding proteins and methods for production.

Claims (24)

1. A method of reducing tumor growth in a subject in need thereof, comprising administering to the subject an effective amount of an isolated monoclonal antibody, which specifically binds to IL-1β, or an antigen binding fragment thereof, wherein said antibody or fragment thereof comprises:

(i) Complementarity Determining Regions (CDRs) according to the Kabat numbering convention of a light chain comprising the amino acid sequence of SEQ ID NO: 17; and

(ii) CDRs according to the Kabat numbering convention of a heavy chain comprising the amino acid sequence of SEQ ID NO: 14.

2. The method of claim 1 , wherein the IL-1β is human, and wherein the antibody or fragment is fully human.

3. The method of claim 2 , wherein the antibody is of the subtype IgG1, IgG2, IgG3 or IgG4.

4. The method of claim 3 , wherein the antibody is of the subtype IgG4.

5. The method of claim 1 , wherein the antibody or fragment is in a composition, and wherein the composition further comprises a pharmaceutically acceptable carrier.

6. A method of reducing tumor growth in a subject in need thereof, comprising administering to the subject an effective amount of an isolated monoclonal antibody which specifically binds to IL-1β, or an antigen binding fragment thereof, wherein said antibody or fragment thereof comprises the following Complementarity Determining Regions (CDRs):

(i) a heavy chain variable region CDR H1 comprising the amino acid sequence of SEQ ID NO:26,

(ii) a heavy chain variable region CDR H2 comprising the amino acid sequence of SEQ ID NO:27,

(iii) a heavy chain variable region CDR H3 comprising the amino acid sequence of SEQ ID NO:28,

(iv) a light chain variable region CDR L1 comprising the amino acid sequence of SEQ ID NO:29,

(v) a light chain variable region CDR L2 comprising the amino acid sequence of SEQ ID NO:30, and

(vi) a light chain variable region CDR L3 comprising an amino acid sequence selected from the group consisting of: SEQ ID NO:12, SEQ ID NO:11, SEQ ID NO:9, SEQ ID NO:10, and SEQ ID NO:13.

7. The method of claim 6 , wherein the light chain variable region CDR L3 comprises the amino acid sequence of SEQ ID NO:12.

8. The method of claim 6 , wherein the light chain variable CDR3 comprises the amino acid sequence of SEQ ID NO:11.

9. The method of claim 6 , wherein the IL-1β is human, and wherein the antibody or fragment is fully human.

10. The method of claim 6 , wherein the antibody is of the subtype IgG1, IgG2, IgG3 or IgG4.

11. A method of reducing tumor growth in a subject in need thereof, comprising administering to the subject an effective amount of an isolated monoclonal antibody which specifically binds to IL-1β, or an antigen binding fragment thereof, wherein said antibody or fragment thereof comprises:

(i) a light chain sequence comprising the amino acid sequence of SEQ ID NO: 17; and

(ii) a heavy chain sequence comprising the amino acid sequence of SEQ ID NO: 18.

12. The method of claim 11 , wherein the heavy chain sequence comprises the amino acid sequence of SEQ ID NO: 14.

13. The method of claim 11 , wherein the IL-1β is human, and wherein the antibody or fragment is fully human.

14. The method of claim 11 , wherein the antibody is of the subtype IgG1, IgG2, IgG3 or IgG4.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 9, 2019
From: WANG, CHENG-I; GOH, ANGELINE; YEO, SIOK PING; MORTELLARO, ALESSANDRA; BISWAS, SUBHRA KUMAR; GINHOUX, FLORENT; ZHONG, PINGYU
To: AGENCY FOR SCIENCE, TECHNOLOGY AND RESEARCH
Reel/Frame 047939/0025 →
Priority Claims (1)
SG 201201007 · Feb 13, 2012 · national
Continuity (2)
Division 14378442
Related Publication 20190144535A1 · May 16, 2019