IP Library Granted Patent US 10,525,095
Granted Patent B2
US 10,525,095 · App. 16/261,773 · Granted Jan 7, 2020

Pharmaceutical composition comprising refined

Inventors: Laurent Chantalat (Antibes, FR); Philippe Andres (Peymeinade, FR)
Assignee: Galderma S.A.
A61K36/70A61K8/492A61K8/4953A61K8/97A61K9/0014A61K9/0053A61K9/06A61K31/404A61K31/519A61K36/19A61K36/315A61K36/48A61Q19/08A61K2236/00A61K2800/92
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Quick Facts
Patent No.
US 10,525,095
App. No.
16/261,773
Granted
Jan 7, 2020
Kind
B2
Abstract

A refined Indigo Naturalis extract or Indigo-producing plant extract containing at least 65% (w/w) an indirubin derivative based on total weight of active ingredients is described. Also described are a pharmaceutical composition containing the refined extract, and the use of the pharmaceutical composition for treating or alleviating a disease or condition.

Claims (16)

1. A method of treating a disease or condition selected from the group consisting of psoriasis, an inflammatory skin condition, onychomycosis, skin cancer, abnormal keratinization induced disease, skin aging, and pustular dermatosis, comprising administering to a subject in need thereof a pharmaceutical composition comprising a solid extract of Indigo Naturalis, wherein the solid extract comprises, relative to the total weight of the extract:

65% to 90% (w/w) indirubin;

0.1-15% (w/w) indigo; and

0.01-5% (w/w) tryptanthrin,

wherein the pharmaceutical composition comprises 0.002% to 0.077% (w/w) of the solid extract relative to the total weight of the pharmaceutical composition.

2. The method of claim 1 , wherein the solid extract comprises 0.1-5% (w/w) tryptanthrin relative to the total weight of the extract.

3. The method of claim 2 , wherein the solid extract further comprises 0.1-5% (w/w) qingdainone relative to the total weight of the extract.

4. The pharmaceutical composition of claim 1 , wherein the solid extract is micronized and comprises particles having a particle size of less than or equal to 30 μm in 99% of the particles.

5. The method of claim 1 , wherein the pharmaceutical composition is orally administered.

6. The method of claim 1 , wherein the pharmaceutical composition is topically administered.

7. The method of claim 1 , wherein the disease or condition is psoriasis, onychomycosis, skin aging, or pustular dermatosis.

8. The method of claim 1 , wherein the disease or condition is the inflammatory skin condition selected from the group consisting of atopic dermatitis (AD), eczema, and superinfected skin.

9. The method of claim 1 , wherein the disease or condition is the skin aging selected from skin rejuvenation, tissue regeneration for scars and skin senescence.

10. The method of claim 1 , wherein the disease or condition is the pustular dermatosis selected from acne, ichthyosis, and palmoplantar keratoderma.

11. The method of claim 1 , wherein the pharmaceutical composition further comprises a pharmaceutically acceptable carrier.

12. The method of claim 11 , wherein the pharmaceutical carrier comprises at least one of an oil, an emulsifier, a thickening agent, and a preservative.

Assignments (3)
MERGER AND CHANGE OF NAME Recorded Mar 10, 2022
From: NESTLÉ SKIN HEALTH SA; GALDERMA HOLDINGS SA
To: GALDERMA HOLDING SA
Reel/Frame 060044/0523 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 10, 2021
From: GALDERMA S.A.
To: NESTLÉ SKIN HEALTH SA
Reel/Frame 058962/0638 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 30, 2019
From: CHANTALAT, LAURENT; ANDRES, PHILIPPE
To: GALDERMA S.A.
Reel/Frame 048192/0281 →