IP Library Patent Application 16274370
Patent Application
App. No. 16/274,370

ACTIVATION OF TRPA1+ NOCICEPTORS IN THE VAGUS NERVE ATTENUATES SYSTEMIC INFLAMMATION

Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US None
App. No.
16/274,370
Abstract

Methods are disclosed for treating inflammation and sepsis and for promoting thermoregulation by activating neurons expressing TRPA1 in the vagus nerve.

Claims (13)

1 . A method of suppressing or ameliorating inflammation, promoting thermoregulation, and/or treating sepsis in a subject comprising activating neurons expressing the ion channel designated transient receptor potential cation channel, subfamily A, member 1 (TRPA1) in the subject's vagus nerve effective to suppress or ameliorate inflammation, promote thermoregulation, and/or treat sepsis in a subject.

2 . The method of claim 1 , wherein TRPA1-positive neurons are activated by administering a TRPA1 nociceptor agonist to the subject.

3 . The method of claim 1 , wherein the method of suppressing inflammation, promoting thermoregulation, and/or treating sepsis is activated by selectively stimulating vagus nerve fibers expressing TRPA1 nociceptors in the subject.

4 . The method of claim 3 , comprising activating vagus nerve afferents.

5 . The method of claim 1 , wherein a photochemical activator is administered to the subject and TRPA1+ nociceptors are activated using optogenetic stimulation.

6 . The method of claim 5 , wherein optovin is administered to the subject and TRPA1+ nociceptors are activated using optogenetic stimulation.

7 . The method of claim 1 , wherein the subject has sepsis.

8 . The method of claim 1 , wherein the subject has endotoxemia, septicemia or septic shock.

9 . The method of claim 1 , wherein activation of TRPA1+ neurons attenuates serum levels of one or more pro-inflammatory cytokines.

10 . The method of claim 9 , wherein activation of TRPA1+ neurons attenuates serum levels of tumor necrosis factor (TNF).

11 . A method of suppressing or ameliorating fever in a subject comprising administering to the subject an antagonist of TRPA1 in amount effective to suppress or ameliorate fever in a subject.

12 . A method of activating an immune response in an immunosuppressed subject comprising administering to the subject an antagonist of TRPA1 in amount effective to induce an immune response in a subject.

13 . The method of claim 1 , wherein the subject is human.

Assignments (5)
CONFIRMATORY LICENSE Recorded Sep 20, 2021
From: EINSTEIN INSTITUTE FOR MEDICAL RESEARCH
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 057531/0516 →
CORRECTIVE ASSIGNMENT TO CORRECT THE 2ND PROPERTY NUMBER PREVIOUSLY RECORDED AT REEL: 050188 FRAME: 0819-0826. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded Nov 10, 2020
From: THE FEINSTEIN INSTITUTE FOR MEDICAL RESEARCH
To: THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH
Reel/Frame 054372/0951 →
CHANGE OF NAME Recorded Aug 27, 2019
From: THE FEINSTEIN INSTITUTE FOR MEDICAL RESEARCH
To: THE FEINSTEIN INSTITUTES FOR MEDICAL RESEARCH
Reel/Frame 050188/0819 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 18, 2019
From: TRACEY, KEVIN J.; CHAVAN, SANGEETA S.; SILVERMAN, HAROLD A.
To: THE FEINSTEIN INSTITUTE FOR MEDICAL RESEARCH
Reel/Frame 048621/0608 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 11, 2019
From: TRACEY, KEVIN J.; CHAVAN, SANGEETA S.; SILVERMAN, HAROLD A.
To: THE FEINSTEIN INTITUTE FOR MEDICAL RESEARCH
Reel/Frame 048556/0446 →