IP Library Granted Patent US 10,842,768
Granted Patent B2
US 10,842,768 · App. 16/364,720 · Granted Nov 24, 2020

Compositions and methods for lowering triglycerides

Inventors: Ian Osterloh (Kent, GB); Pierre Wicker (Mystic, CT); Rene Braeckman (Richboro, PA); Paresh Soni (Mystic, CT); Mehar Manku (Birmingham, GB)
Assignee: Amarin Pharmaceuticals Ireland Limited
A61K31/232A61K9/48A61K31/202A61K31/366A61K31/40A61K31/505A61P9/10
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Quick Facts
Patent No.
US 10,842,768
App. No.
16/364,720
Granted
Nov 24, 2020
Kind
B2
Abstract

In various embodiments, the present invention provides compositions and methods for treating and/or preventing cardiovascular-related diseases in subject in need thereof.

Claims (9)

1. A method of lowering triglycerides and LDL-C in a subject comprising, administering orally to a subject having fasting triglycerides of about 200 mg/dl to less than 500 mg/dl who is on stable statin therapy about 4 g per day of a pharmaceutical composition comprising at least about 96%, by weight of all fatty acids present, ethyl eicosapentaenoate for a period of at least about 12 weeks to effect a reduction in fasting triglycerides and fasting LDL-C in the subject, wherein the stable statin therapy comprises administering about 10 mg to about 100 mg per day of a statin selected from atorvastatin, rosuvastatin and simvastatin.

2. The method of claim 1 , comprising administering the composition to effect a reduction in fasting non-HDL-C.

3. The method of claim 1 , comprising administering the composition to effect a reduction in fasting VLDL-C.

4. The method of claim 1 , comprising administering the composition to effect a reduction in fasting Apolipoprotein B.

5. The method of claim 1 , comprising administering the composition to effect a reduction in fasting total cholesterol.

6. A method of lowering triglycerides and LDL-C in a subject comprising, administering orally to a subject having fasting triglycerides from about 200 mg/dl to less than 500 mg/dl who is on stable statin therapy about 4 g per day of a pharmaceutical composition comprising at least about 96%, by weight of all fatty acids present, ethyl eicosapentaenoate for a period of at least about 12 weeks to effect a reduction in fasting triglycerides in the subject by least 5% and to effect a reduction in fasting LDL-C in the subject by at least about 5%, wherein the stable statin therapy comprises administering about 10 mg to about 100 mg per day of a statin selected from atorvastatin, rosuvastatin and simvastatin.

7. The method of claim 6 , comprising administering the composition to effect at least a 5% reduction in fasting LDL-C.

8. A method of lowering triglycerides in a subject on stable statin therapy and having fasting a baseline triglyceride level from about 200 mg/dl to less than 500 mg/dl comprising administering orally to the subject about 4 g per day of a pharmaceutical composition comprising at least about 96%, by weight of all fatty acids present, ethyl eicosapentaenoate for a period of 12 weeks, which when administered to a first patient population on stable statin therapy and having said baseline triglyceride level at 4 g per day for twelve weeks is effective to reduce fasting triglycerides and fasting LDL-C, wherein the stable statin therapy comprises about 10 mg to about 100 mg per day of a statin selected from atorvastatin, rosuvastatin and simvastatin.

9. The method of claim 6 , comprising administering the composition to effect a reduction in fasting non-HDL-C.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 8, 2019
From: OSTERLOH, IAN; WICKER, PIERRE; BRAECKMAN, RENE; SONI, PARESH; MANKU, MEHAR
To: AMARIN PHARMA, INC.
Reel/Frame 049692/0565 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 8, 2019
From: AMARIN PHARMA, INC.
To: AMARIN PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 049692/0576 →