IP Library Granted Patent US 10,912,783
Granted Patent B2
US 10,912,783 · App. 16/401,884 · Granted Feb 9, 2021

Formulations for solubilizing hormones

Inventors: Thorsteinn Thorsteinsson (Boynton Beach, FL); Frederick D. Sancilio (Palm Beach Gardens, FL); Brian A. Bernick (Boca Raton, FL); Julia M. Amadio (Boca Raton, FL)
Assignee: THERAPEUTICSMD, INC.
A61K31/573A61K9/0014A61K9/06A61K9/4825A61K9/4858A61K31/015A61K31/565A61K47/06A61K47/14
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Quick Facts
Patent No.
US 10,912,783
App. No.
16/401,884
Granted
Feb 9, 2021
Kind
B2
Abstract

Compositions and methods for the solubilization of steroid hormones are disclosed.

Claims (6)

1. A liquid composition comprising about 100 mg progesterone- and d-limonene; wherein the progesterone and d-limonene are present in a weight ratio that does not exceed 1 part progesterone to 4.9 parts d-limonene, further wherein the liquid composition is encapsulated in a soft gelatin capsule suitable for oral administration; and wherein the progesterone is micronized.

2. The liquid composition of claim 1 , further comprising an antioxidant.

3. The liquid composition of claim 2 , wherein the antioxidant is selected from the group consisting of α-tocopherol acetate, acetone sodium bisulfite, acetyl cysteine, ascorbic acid, ascorbyl palmitate, butylated hydroxyanisole (BHA), butylated hydroxytoluene (BHT), cysteine, cysteine hydrochloride, α-tocopherol, dithiothreitol, monothioglycerol, nordihydroguaiaretic acid, propyl gallate, sodium bisulfite, sodium formaldehyde sulfoxylate, sodium metabisulfite, sodium sulfite, sodium thiosulfate, thiourea, tocopherol, and combinations thereof.

4. The liquid composition of claim 1 , wherein the composition comprises at least about 80% w/w d-limonene.

5. The liquid composition of claim 4 , further comprising an antioxidant.

6. The liquid composition of claim 1 further comprising estradiol.

Assignments (6)
TERMINATION AND RELEASE OF GRANT OF A SECURITY INTEREST - PATENTS Recorded Dec 30, 2022
From: SIXTH STREET SPECIALTY LENDING, INC. (F/K/A TPG SPECIALTY LENDING, INC.)
To: THERAPEUTICSMD, INC.
Reel/Frame 062254/0813 →
CORRECTIVE ASSIGNMENT TO CORRECT THE APPLICATION NO. 16/401,844 PREVIOUSLY RECORDED AT REEL: 050928 FRAME: 0987. ASSIGNOR(S) HEREBY CONFIRMS THE CHANGE OF ADDRESS. Recorded Sep 24, 2021
From: THERAPEUTICSMC, INC.
To: THERAPEUTICSMD, INC.
Reel/Frame 057698/0571 →
SECURITY INTEREST Recorded Jan 27, 2021
From: THERAPEUTICSMD, INC.
To: SIXTH STREET SPECIALTY LENDING, INC. (F/K/A TPG SPECIALTY LENDING, INC.)
Reel/Frame 055049/0651 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2020
From: AMADIO, JULIA M.; BERNICK, BRIAN A.
To: THERAPEUTICSMD, INC.
Reel/Frame 054151/0543 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 15, 2020
From: SANCILIO, FREDERICK D.; THORSTEINSSON, THORSTEINN
To: THERAPEUTICSMD, INC.
Reel/Frame 054067/0602 →
CHANGE OF ADDRESS Recorded Nov 5, 2019
From: THERAPEUTICSMD, INC.
To: THERAPEUTICSMD, INC.
Reel/Frame 050928/0987 →
Continuity (3)
Division 15217301 · Jul 22, 2016
Provisional Application 62196021 · Jul 23, 2015
Related Publication 20190321376A1 · Oct 24, 2019