IP Library Granted Patent US 10,676,471
Granted Patent B2
US 10,676,471 · App. 16/416,997 · Granted Jun 9, 2020

Cycloalkyl-linked diheterocycle derivatives

Inventors: Aaron Craig Burns (San Diego, CA); Michael Raymond Collins (San Diego, CA); Samantha Elizabeth Greasley (San Diego, CA); Robert Louis Hoffman (Carlsbad, CA); Peter Qinhua Huang (San Diego, CA); Robert Steven Kania (Solana Beach, CA); Pei-Pei Kung (San Diego, CA); Maria Angelica Linton (San Diego, CA); Lakshmi Sourirajan Narasimhan (San Diego, CA); Paul Francis Richardson (San Diego, CA); Daniel Tyler Richter (San Diego, CA); Graham Smith (San Diego, CA)
Assignee: Pfizer Inc.
C07D417/14C07D417/08A61K31/427A61K31/444A61K31/4439A61K31/501A61K31/506A61K45/06C07D277/46C07D401/14
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Quick Facts
Patent No.
US 10,676,471
App. No.
16/416,997
Granted
Jun 9, 2020
Kind
B2
Abstract

The present invention relates to compounds of formula (I) or pharmaceutically acceptable salts thereof, wherein A, L, D, R 1 -R 15 , w, x, y, and z are defined herein. The novel cycloalkyl-linked diheterocycle derivatives that are useful in the treatment of abnormal cell growth, such as cancer, in mammals. The present invention also relates to pharmaceutical compositions containing the compounds and to methods of using the compounds and compositions in the treatment of abnormal cell growth in mammals.

Claims (3)

1. A compound selected from the group consisting of

or a pharmaceutically acceptable salt thereof.

2. A pharmaceutical formulation comprising at least one compound of claim 1 , or a pharmaceutically acceptable salt thereof, and at least one pharmaceutically acceptable carrier, diluent, or excipient.

Assignments (1)
ASSIGNEE ADDRESS CORRECTION Recorded Mar 20, 2023
From: PFIZER INC.
To: PFIZER INC.
Reel/Frame 063119/0087 →