IP Library Granted Patent US 10,722,478
Granted Patent B2
US 10,722,478 · App. 16/537,170 · Granted Jul 28, 2020

Methods and compositions for treating fatigue associated with disordered sleep using very low dose cyclobenzaprine

Inventors: Seth Lederman (New York, NY); Herb Harris (Chapel Hill, NC)
Assignee: Tonix Pharma Holdings Limited
A61K31/135A61K9/0053A61K9/2018A61K9/2059A61K9/28A61K9/4825A61K31/137A61K45/06G16C99/00A61K9/2866
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Quick Facts
Patent No.
US 10,722,478
App. No.
16/537,170
Granted
Jul 28, 2020
Kind
B2
Abstract

The present invention relates to methods for the treatment or prevention of fatigue associated with disordered sleep, for example, in multiple sclerosis, fibromyalgia, Fabry's disease, Parkinson's disease, or traumatic brain injury, using cyclobenzaprine. The present invention further relates to a biomarker for the therapeutic effects of a cyclobenzaprine treatment.

Claims (5)

1. A method for reducing CAP rates A2 or A3, comprising administering to a human in need of such treatment a pharmaceutical composition comprising cyclobenzaprine and a pharmaceutically acceptable carrier, wherein such treatment reduces CAP rates A2 or A3, and wherein the amount of cyclobenzaprine administered is less than 5 mg/day.

2. The method of claim 1 , wherein the amount of cyclobenzaprine administered is less than 2.5 mg/day.

3. The method of claim 1 , wherein the method further comprises administering sequentially or concurrently a drug selected from the group consisting of a dual reuptake inhibitor, a serotonin-norepinephrine reuptake inhibitor or a calcium channel inhibitor.

4. The method of claim 1 , wherein the pharmaceutical composition is administered as an orally dissolving tablet, as a thin film formulation, or as a promicellar formulation.

5. The method of claim 1 , wherein the pharmaceutical composition is administered at bedtime.

Assignments (3)
NOVATION AGREEMENT Recorded Sep 25, 2024
From: TONIX PHARMA HOLDINGS LIMITED
To: TONIX PHARMA LIMITED
Reel/Frame 069504/0760 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 12, 2019
From: LEDERMAN, SETH; HARRIS, HERB
To: TONIX PHARMACEUTICALS, INC.
Reel/Frame 050023/0488 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 12, 2019
From: TONIX PHARMACEUTICALS, INC.
To: TONIX PHARMA HOLDINGS LIMITED
Reel/Frame 050023/0511 →
Continuity (5)
Continuation 15266035 · Sep 15, 2016
Division 14477981 · Sep 5, 2014
Division 13157270 · Jun 9, 2011
Provisional Application 61358305 · Jun 24, 2010
Related Publication 20190358177A1 · Nov 28, 2019