IP Library Granted Patent US 11,459,368
Granted Patent B2
US 11,459,368 · App. 16/630,322 · Granted Oct 4, 2022

Insulin-transferrin fusion protein and its prodrug, proinsulin-transferrin, for overcoming insulin resistance

Inventors: Wei-Chiang Shen (San Marino, CA); Yuqian Liu (Henan, CA); Hsuan-Yao Wang (Fullerton, CA)
Assignee: Livactus, Inc.
C07K14/62A61P3/00C07K14/79A61K38/00C07K2319/00
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Quick Facts
Patent No.
US 11,459,368
App. No.
16/630,322
Granted
Oct 4, 2022
Kind
B2
Abstract

A method of treating Type 2 diabetes (T2D) is provided. The method includes administering to a subject in need thereof an effective amount of a pharmaceutical composition that includes an insulin-transferrin fusion protein or its prodrug, proinsulin-transferrin fusion protein.

Claims (9)

1. A method of treating insulin resistance in a subject with diabetes having insulin resistance comprising administering a fusion protein of proinsulin and transferrin (ProINS-Tf) or insulin and transferrin (INS-Tf) to a subject in need thereof in a pharmaceutically acceptable carrier in an effective amount to reduce blood glucose levels in the subject, thereby treating insulin resistance in the subject.

2. The method of claim 1 , wherein the subject was at least partially resistant to insulin prior to treatment.

3. The method of claim 1 , wherein the subject's blood glucose level is at a level of a non-diabetic subject after treatment.

4. The method of claim 3 , wherein glucose levels are reduced within about 4-8 hours of administration.

5. The method of claim 1 , wherein administration is in single-dosage form.

6. The method of claim 1 , further comprising administering a second insulin drug.

7. The method of claim 1 , wherein the subject is a human.

8. A method of treating a subject with insulin resistance comprising administering a fusion protein encoded by a nucleic acid sequence comprising a pre-proinsulin nucleic acid sequence operably linked to a transferrin (Tf) sequence to a subject in need thereof in a pharmaceutically acceptable carrier thereby treating the insulin resistance.

9. The method of claim 1 or 8 , wherein the subject has Type 2 Diabetes (T2D).

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 13, 2022
From: SHEN, WEI-CHIANG; LIU, YUQIAN; WANG, HSUAN-YAO
To: LIVACTUS, INC.
Reel/Frame 059906/0783 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 19, 2021
From: UNIVERSITY OF SOUTHERN CALIFORNIA
To: SHEN, WEI-CHIANG; LIU, YUQIAN; WANG, HSUAN-YAO
Reel/Frame 057235/0224 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 18, 2021
From: SHEN, WEI-CHIANG; LIU, YUQIAN; WANG, HSUAN-YAO
To: UNIVERSITY OF SOUTHERN CALIFORNIA
Reel/Frame 055951/0596 →
Continuity (2)
Provisional Application 62532822 · Jul 14, 2017
Related Publication 20200165315A1 · May 28, 2020