IP Library Granted Patent US 12,392,785
Granted Patent B2
US 12,392,785 · App. 16/635,093 · Granted Aug 19, 2025

Adjusted multi-biomarker disease activity score for inflammatory disease assessment

Inventors: Ching Chang Hwang (South San Francisco, CA); David Chernoff (South San Francisco, CA); Alexander Gutin (Salt Lake City, UT); Darl Flake (Salt Lake City, UT); Jerry Lanchbury (Salt Lake City, UT); Paul Scott Eastman (South San Francisco, CA); Eric Sasso (South San Francisco, CA)
Assignee: LABORATORY CORPORATION OF AMERICA HOLDINGS
G01N33/6893G01N2800/52G01N2800/60G01N2800/7095
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 12,392,785
App. No.
16/635,093
Granted
Aug 19, 2025
Kind
B2
Abstract

Provided herein are methods for assessing response to inflammatory disease therapy. The methods include performing immunoassays to generate scores based on quantitative data for expression of biomarkers relating to inflammatory biomarkers to assess disease activity in inflammatory diseases, e.g., rheumatoid arthritis. Also provided are methods of adjusting disease activity scores to account for variables that can influence such scores.

Claims (15)

1. A method for assessing a subject for treatment for rheumatoid arthritis disease activity, the method comprising:

obtaining a blood sample from the subject;

performing an immunoassay to measure protein expression values of at least six protein markers in the sample, the at least six markers comprising chitinase 3-like 1 (cartilage glycoprotein-39) (CHI3L1), interleukin 6 (interferon, beta 2) (IL6), leptin (LEP), matrix metallopeptidase 1 (interstitial collagenase) (MMP1), matrix metallopeptidase 3 (stromelysin 1, progelatinase) (MMP3), and serum amyloid Al (SAA1);

generating a multi-biomarker disease activity (MBDA) score by (a) weighting the determined expression of each protein marker with a predefined coefficient, and (b) combining the weighted expression; and

calculating a disease activity score for the subject according to the formula:

disease activity score=MBDA score+33.9−{+0.437×age+3.31×1male(sex)+0.0502×leptin 0.58 −0.0247×age×1male(sex)−0.000483×age×leptin 0.58 +0.00254×1male (sex)×leptin 0.58 };

wherein the values+0.437, +3.31, +0.0502,−0.0247,−0.000483, and +0.00254 are stated to a 95% Confidence Interval;

wherein age is the subject's age;

wherein leptin is the subject's leptin value; and

wherein 1male (sex) is 1 for a male subject and is zero otherwise;

determining that the subject has a disease activity score of 45 to 100 and a high level of rheumatoid arthritis disease activity; and

administering a DMARD or biologic DMARD therapy to the subject having a disease activity score of 45 to 100 and a high level of rheumatoid arthritis disease activity.

2. The method of claim 1 , wherein the protein markers further comprise an additional protein marker comprising at least one of C-reactive protein pentraxin-related (CRP), epidermal growth factor (beta-urogastrone) (EGF), resistin (RETN), tumor necrosis factor receptor superfamily, member 1A (TNFRSF1A), vascular cell adhesion molecule 1 (VCAM1), and vascular endothelial growth factor A (VEGFA).

3. The method of claim 2 , wherein the at least one additional protein marker is CRP.

4. The method of claim 2 , wherein the disease activity score is calculated using markers comprising IL6, EGF, VEGFA, LEP, SAA1, VCAMI, CRP, MMP1, MMP3, TNFRSF1A, RETN, and CHI3L1.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 6, 2021
From: CRESCENDO BIOSCIENCE, INC.
To: LABORATORY CORPORATION OF AMERICA HOLDINGS
Reel/Frame 057709/0825 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 2, 2021
From: FLAKE, DARL; GUTIN, ALEXANDER; LANCHBURY, JERRY; CHERNOFF, DAVID; EASTMAN, PAUL SCOTT; SASSO, ERIC; HWANG, CHING CHANG
To: MYRIAD GENETICS, INC.
Reel/Frame 057057/0253 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 14, 2021
From: MYRIAD GENETICS, INC.
To: CRESCENDO BIOSCIENCE, INC.
Reel/Frame 056246/0689 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 25, 2021
From: GUTIN, ALEXANDER; FLAKE, DARL; LANCHBURY, JERRY
To: MYRIAD GENETICS, INC.
Reel/Frame 055417/0620 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 25, 2021
From: HWANG, CHING CHANG; CHERNOFF, DAVID; EASTMAN, PAUL SCOTT; SASSO, ERIC
To: CRESCENDO BIOSCIENCE
Reel/Frame 055417/0704 →
Continuity (3)
Provisional Application 62558413 · Sep 14, 2017
Provisional Application 62538959 · Jul 31, 2017
Related Publication 20200249243A1 · Aug 6, 2020
References Cited (29)
US 20110137851A1 · Cavet · 2011 [cited by examiner]
US 20140057833A1 · Otvos et al. · 2014 [cited by applicant]
US 20140142861A1 · Hagstrom · 2014 [cited by examiner]
JP 2001512482A · 2001 [cited by applicant]
WO 2015191423A1 · 2015 [cited by applicant]
WO 2015191613A1 · 2015 [cited by applicant]
WO 2017058999A2 · 2017 [cited by applicant]
WO 2017059003A1 · 2017 [cited by applicant]
WO 2020186007 · 2020 [cited by applicant]
Bakker; Marije. 2011. Tight control and long-term prediction in rheumatoid arthritis. Research Gate (Year: 2011). [cited by examiner]
Centola, Michael. Development of a Multibiomarker Disease activity test for Rheumatoid arthritis. Plos One. 2013 (Year: 2013). [cited by examiner]
Hambardzumyan, and NPL reference titled Pretreatment multi-biomarker disease activity score and radiographic. 2014 (Year: 2014). [cited by examiner]
Centola et al. , “Development of a multi-biomarker disease activity test for rheumatoid arthritis”, PLoS One. Apr. 9, 2013;8(4):e60635. doi: 10.1371/journal.pone.0060635. [cited by applicant]
Chen et al., “Association between inflammation and insulin resistance in U.S. nondiabetic adults: results from the Third National Health and Nutrition Examination Survey”, Diabetes Care. Dec. 2004;27(12):2960-5. doi: 10… [cited by applicant]
Curtis et al., Development of an adjusted multi-biomarker disease activity (MBDA) score for rheumatoid arthritis (RA) that accounts for age, sex and adiposity, with subsequent evaluation of ability to predict risk for r… [cited by applicant]
Curtis et al., “Adjustment of the multi-biomarker disease activity score to account for age, sex and adiposity in patients with rheumatoid arthritis”, Rheumatology (Oxford). May 1, 2019;58(5):874-883. doi: 10.1093/rheum… [cited by applicant]
Curtis et al., “Influence of obesity, age, and comorbidities on the multi-biomarker disease activity test in rheumatoid arthritis”, Semin Arthritis Rheum. Feb. 2018;47(4):472-477. doi: 10.1016/j.semarthrit.2017.07.010. … [cited by applicant]
Extended European Search Report issued in EP 18840827.2 on Apr. 9, 2021 (17 pages). [cited by applicant]
Hambardzumyan et al., “Pretreatment multi-biomarker disease activity score and radiographic progression in early RA: results from the SWEFOT trial”, Ann Rheum Dis. Jun. 2015;74(6):1102-9. doi: 10.1136/annrheumdis-2013-2… [cited by applicant]
Kitahara et al., “Body mass index, physical activity, and serum markers of inflammation, immunity, and insulin resistance”, Cancer Epidemiol Biomarkers Prev. Dec. 2014;23(12):2840-9. doi: 10.1158/1055-9965.EPI-14-0699-T… [cited by applicant]
Ranganath et al., “Age adjustment corrects for apparent differences in erythrocyte sedimentation rate and C-reactive protein values at the onset of seropositive rheumatoid arthritis in younger and older patients”, J Rhe… [cited by applicant]
International Search Report issued in PCT/US2018/044396 on Mar. 4, 2019 (4 pages). [cited by applicant]
Lee et al., “Measurement of the serum leptin level could assist disease activity monitoring in rheumatoid arthriti”, Rheumatol Int. Apr. 2007;27(6):537-40. Epub Nov. 11, 2006. (Abstract only). [cited by applicant]
Curtis et al, “Validation of a novel multibiomarker test to assess rheumatoid arthritis disease activity”, Arthritis Care Res (Hoboken). Dec. 2012;64(12):1794-803. doi: 10.1002/acr.21767. [cited by applicant]
Japanese Patent Application No. 2020-505174, Office Action mailed Jun. 21, 2022, 12 pages. [cited by applicant]
Japanese Patent Application No. 2020-505174, Office Action mailed Aug. 29, 2023, 5 pages. [cited by applicant]
Japanese Patent Application No. P2020-505174, Office Action mailed Apr. 11, 2023, 6 pages. [cited by applicant]
Canadian Patent Application No. 3,071,597, Office Action mailed on Jul. 29, 2024, 4 pages. [cited by applicant]
European Patent Application No. 18840827.2, Office Action mailed on Jul. 15, 2024, 10 pages. [cited by applicant]