IP Library Granted Patent US 11,020,385
Granted Patent B2
US 11,020,385 · App. 16/730,015 · Granted Jun 1, 2021

Combination therapy

Inventors: Casey Kopczynski (Chapel Hill, NC); Cheng-Wen Lin (Raleigh, NC); Jill Marie Sturdivant (Chapel Hill, NC); Mitchell A. deLong (Chapel Hill, NC)
Assignee: Aerie Pharmaceuticals, Inc.
A61K31/472A61K9/0048A61K9/08A61K31/4725A61K31/557A61K31/559A61K31/5575A61K47/54A61K47/55C07D217/22C07D409/12
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Quick Facts
Patent No.
US 11,020,385
App. No.
16/730,015
Granted
Jun 1, 2021
Kind
B2
Abstract

Described herein are compounds and compositions for treating glaucoma and/or reducing intraocular pressure. Compositions may comprise an isoquinoline compound and a prostaglandin or a prostaglandin analog. Compounds described herein include those in which an isoquinoline compound is covalently linked to a prostaglandin or a prostaglandin analog, and those in which an isoquinoline compound and a prostaglandin free acid together form a salt.

Claims (10)

1. A method of treating glaucoma or ocular hypertension, comprising administration via ocular instillation of a composition comprising a Rho kinase inhibitor and a pharmaceutically acceptable carrier to a subject in need thereof,

wherein the administration is daily administration,

wherein the Rho kinase inhibitor is (S)-4-(3-amino-1-(isoquinolin-6-ylamino)-1-oxopropan-2-yl)benzyl 2,4-dimethylbenzoate dimesylate.

2. The method of claim 1 , wherein the administration is daily administration for up to one year.

3. The method of claim 1 , wherein the amount of the Rho kinase inhibitor administered is about one drop of an about 0.02% solution of the Rho kinase inhibitor per eye of the subject.

4. The method of claim 2 , wherein the amount of the Rho kinase inhibitor administered is about one drop of an about 0.02% solution of the Rho kinase inhibitor per eye of the subject.

5. The method of claim 1 , wherein the daily administration is once daily.

6. The method of claim 2 , wherein the daily administration is once daily.

7. The method of claim 3 , wherein the daily administration is once daily.

8. The method of claim 4 , wherein the daily administration is once daily.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 24, 2024
From: AERIE PHARMACEUTICALS, INC.
To: ALCON INC.
Reel/Frame 067822/0168 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 30, 2019
From: KOPCZYNSKI, CASEY; LIN, CHENG-WEN; STURDIVANT, JILL MARIE; DELONG, MITCHELL A.
To: AERIE PHARMACEUTICALS, INC.
Reel/Frame 051386/0403 →