IP Library Granted Patent US 11,497,750
Granted Patent B2
US 11,497,750 · App. 16/804,092 · Granted Nov 15, 2022

Methods of treating and/or preventing actinic keratosis

Inventors: Min-Fun Rudolf Kwan (Summit, NJ); Johnson Yiu-Nam Lau (Houston, TX); E. Douglas Kramer (Stamford, CT); David Lawrence Cutler (Moorestown, NJ); Jane Fang (Newport Beach, CA)
Assignee: ATNX SPV, LLC
A61K31/5377A61K9/0014A61P17/00
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Quick Facts
Patent No.
US 11,497,750
App. No.
16/804,092
Granted
Nov 15, 2022
Kind
B2
Abstract

The application pertains to methods of treating and/or preventing actinic keratosis, comprising administering a therapeutically effective amount of KX-01, to a subject in need thereof.

Claims (24)

1. A method of treating actinic keratosis comprising administering to a subject in need thereof a compound of the following structure:

at dose from about 0.1 mg to about 10 mg, to an affected area of the subject.

2. The method of claim 1 , wherein the affected area is about 0.01 cm 2 to about 300 cm 2 .

3. The method of claim 1 , wherein the affected area is about 10 cm 2 to about 200 cm 2 .

4. The method of claim 1 , wherein the affected area is the skin.

5. The method of claim 1 , wherein the affected area is about 25 cm 2 .

6. The method of claim 1 , wherein the affected area is about 100 cm 2 .

7. The method of claim 1 , wherein the subject has one affected area.

8. The method of claim 1 , wherein the subject has more than one affected area.

9. The method of claim 1 , wherein the compound is administered once a week, once every three days, once every two days, once a day, twice a day, three times a day, or four times a day.

10. The method of claim 1 , wherein the compound is administered for 1, 2, 3, 4, or 5 days.

11. The method of claim 1 , wherein the compound is administered for 1, 2, 3, 4, 5, or 6 days per week.

12. The method of claim 1 , wherein the compound is administered once or twice daily continuously for more than one day per week, followed by discontinuation of the administration for the rest of the week.

13. The method of claim 1 , wherein the compound is administered topically.

14. The method of claim 1 , wherein the treatment comprises reducing the number and/or severity of, or the number of the subjects that have, local skin reactions or other adverse side effects in the subject compared to other treatments of actinic keratosis.

15. The method of claim 1 , wherein the compound is administered to an affected area of the subject at a dose from about 0.2 mg to about 5 mg.

16. The method of claim 1 , wherein the compound is administered to an affected area of the subject at a dose from about 0.5 mg to about 2.5 mg.

17. The method of claim 15 , wherein the compound is administered to an affected area of the subject at a dose of about 0.2 mg, about 0.3 mg, about 0.4 mg, about 0.5 mg, about 0.6 mg, about 0.7 mg, about 0.8 mg, about 0.9 mg, about 1 mg, about 1.1 mg, about 1.2 mg, about 1.3 mg, about 1.4 mg, about 1.5 mg, about 1.6 mg, about 1.7 mg, about 1.8 mg, about 1.9 mg, about 2.0 mg, about 2.1 mg, about 2.2 mg, about 2.3 mg, about 2.4 mg, about 2.5 mg, about 2.6 mg, about 2.7 mg, about 2.8 mg, about 2.9 mg, about 3 mg, about 4 mg, or about 5 mg.

18. The method of claim 16 , wherein the compound is administered to an affected area of the subject at a dose of about 0.5 mg, about 0.6 mg, about 0.7 mg, about 0.8 mg, about 0.9 mg, about 1 mg, about 1.1 mg, about 1.2 mg, about 1.3 mg, about 1.4 mg, about 1.5 mg, about 1.6 mg, about 1.7 mg, about 1.8 mg, about 1.9 mg, about 2.0 mg, about 2.1 mg, about 2.2 mg, about 2.3 mg, about 2.4 mg, or about 2.5 mg.

19. The method of claim 1 , wherein the compound is administered once daily.

20. The method of claim 1 , wherein the compound is administered for 3 days.

21. The method of claim 1 , wherein the compound is administered for 5 days.

22. The method of claim 1 , wherein the compound is administered at a dose of about 0.5 mg once daily for 3 days.

23. The method of claim 1 , wherein the compound is administered at a dose of about 0.5 mg once daily for 5 days.

Assignments (5)
SECURITY INTEREST Recorded Sep 16, 2022
From: ATHENEX, INC.
To: SAGARD HEALTHCARE ROYALTY PARTNERS, LP, AS ADMINISTRATIVE AGENT
Reel/Frame 061119/0681 →
SECURITY INTEREST Recorded Sep 16, 2022
From: ATNX SPV, LLC
To: SAGARD HEALTHCARE ROYALTY PARTNERS, LP, AS ADMINISTRATIVE AGENT
Reel/Frame 061119/0920 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 13, 2022
From: ATHENEX, INC.
To: ATNX SPV, LLC
Reel/Frame 061071/0086 →
SECURITY INTEREST Recorded Jun 22, 2020
From: ATHENEX, INC.
To: OAKTREE FUND ADMINISTRATION, LLC
Reel/Frame 053005/0657 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 28, 2020
From: KWAN, MIN-FUN RUDOLF; LAU, JOHNSON YIU-NAM; KRAMER, E. DOUGLAS; CUTLER, DAVID LAWRENCE; FANG, JANE
To: ATHENEX, INC.
Reel/Frame 051958/0772 →
Continuity (3)
Continuation 15918100 · Mar 12, 2018
Provisional Application 62469889 · Mar 10, 2017
Related Publication 20200197405A1 · Jun 25, 2020
Cited By (1)
US 12,215,083