IP Library Granted Patent US 11,021,481
Granted Patent B2
US 11,021,481 · App. 17/020,173 · Granted Jun 1, 2021

Substituted isoindolin-1-ones and 2,3-dihydro-1h-pyrrolo[3,4-c]pyridin-1-ones as HPK1 antagonists

Inventors: Neelu Kaila (Lexington, MA); Ian Linney (Saffron Walden, GB); Stuart Ward (Saffron Walden, GB); Grant Wishart (Saffron Walden, GB); Ben Whittaker (Saffron Walden, GB); Alexandre Cote (West New York, NJ); Jeremy Robert Greenwood (Brooklyn, NY); Abba Leffler (Bronx, NY); Steven K. Albanese (Brooklyn, NY); Daniel L. Severance (San Diego, CA)
Assignee: Nimbus Saturn, Inc.
C07D471/04C07D519/00
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Quick Facts
Patent No.
US 11,021,481
App. No.
17/020,173
Granted
Jun 1, 2021
Kind
B2
Abstract

The present invention provides compounds, compositions thereof, and methods of using the same for the inhibition of HPK1, and the treatment of HPK1-mediated disorders.

Claims (44)

1. A compound selected from the group consisting of:

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

3. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

4. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

5. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

6. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

7. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

8. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

9. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

10. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

11. The compound of claim 1 , wherein said compound is

or a pharmaceutically acceptable salt thereof.

12. A pharmaceutical composition comprising a compound selected from the group consisting of:

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

13. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

14. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

15. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

16. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

17. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

18. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

19. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

20. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

21. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

22. The pharmaceutical composition of claim 12 , wherein said compound is

or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable carrier, adjuvant, or vehicle.

Assignments (15)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: WISHART, GRANT
To: CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Reel/Frame 055981/0730 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: KAILA, NEELU
To: NIMBUS DISCOVERY, INC.
Reel/Frame 055156/0036 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: WHITTAKER, BEN
To: CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Reel/Frame 055156/0219 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: COTE, ALEXANDRE
To: SCHRÖDINGER, INC.
Reel/Frame 055156/0224 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: GREENWOOD, JEREMY ROBERT
To: SCHRÖDINGER, INC.
Reel/Frame 055156/0229 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: LEFFLER, ABBA
To: SCHRÖDINGER, INC.
Reel/Frame 055156/0238 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: ALBANESE, STEVEN K.
To: SCHRÖDINGER, INC.
Reel/Frame 055156/0246 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: SEVERANCE, DANIEL L.
To: SCHRÖDINGER, INC.
Reel/Frame 055156/0261 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: CHARLES RIVER LABORATORIES, INC.
To: NIMBUS DISCOVERY, INC.
Reel/Frame 055156/0283 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: SCHRÖDINGER, INC.
To: SCHRÖDINGER, L.L.C.
Reel/Frame 055156/0301 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: SCHRÖDINGER, L.L.C.
To: NIMBUS DISCOVERY, INC.
Reel/Frame 055156/0315 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: NIMBUS DISCOVERY, INC.
To: NIMBUS SATURN, INC.
Reel/Frame 055156/0335 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: LINNEY, IAN
To: CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LTD.
Reel/Frame 055223/0911 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: WARD, STUART
To: CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
Reel/Frame 055223/0928 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 4, 2021
From: CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED
To: CHARLES RIVER LABORATORIES, INC.
Reel/Frame 055224/0079 →
Continuity (4)
Continuation 17018591 · Sep 11, 2020
Provisional Application 63032070 · May 29, 2020
Provisional Application 62900152 · Sep 13, 2019
Related Publication 20210087190A1 · Mar 25, 2021
Cited By (3)
US 12,215,105 US 12,252,488 US 12,466,841