IP Library Granted Patent US 12,364,687
Granted Patent B2
US 12,364,687 · App. 17/056,559 · Granted Jul 22, 2025

Use of riluzole oral disintegrating tablets for treating diseases

Inventors: Vladimir Coric (Madison, CT); Robert Berman (New Haven, CT); Irfan Qureshi (Hackensack, NJ)
Assignee: Biohaven Therapeutics Ltd.
A61K31/428A61K9/0056A61K9/006A61K9/2018A61K9/2063A61K9/2095A61P21/00A61P25/28
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Quick Facts
Patent No.
US 12,364,687
App. No.
17/056,559
Granted
Jul 22, 2025
Kind
B2
Abstract

Disclosed are methods of treating a disease in a patient in need thereof, comprising administering to the patient a pharmaceutical composition comprising a therapeutically effective amount of riluzole, or a pharmaceutically acceptable salt thereof, in the form of an oral solid molded fast-dispersing dosage form. Pharmaceutical compositions and kits are also disclosed.

Claims (4)

1. A method of treating cerebellar ataxia in a patient in need thereof, comprising administering to the patient a pharmaceutical composition comprising 50-70% riluzole, 15-25 weight % gelatin, 10-20 weight % mannitol, and 0.1-2 weight % docusate sodium, based on the total weight of the pharmaceutical composition, in the form of an oral solid molded fast-dispersing dosage form in order to provide an AUC 0-t of from about 80-125% of about 740000 hr*pg/mL, wherein the dosage of riluzole in the oral solid molded fast dispersing tablet is from 50 to 90% of the dosage of riluzole in a conventional tablet in order to provide an AUC 0-t of about 740000 hr*pg/mL.

2. The method of claim 1 , wherein the dosage of riluzole in the oral solid molded fast dispersing tablet is from 70 to 85% of the dosage of riluzole in a conventional tablet in order to provide an AUC 0-t of about 740000 hr*pg/mL.

3. The method of claim 2 , wherein the dosage of riluzole in the oral solid molded fast dispersing tablet is about 80% of the dosage of riluzole in a conventional tablet in order to provide an AUC 0-t of about 740000 hr*pg/mL.

4. The method of claim 1 , wherein the dosage of riluzole in the oral solid molded fast dispersing tablet is about 40 mg.

Assignments (2)
RELEASE OF SECURITY INTEREST Recorded Apr 27, 2025
From: SIXTH STREET SPECIALTY LENDING, INC.
To: BIOHAVEN PHARMACEUTICAL HOLDING COMPANY LTD.; BIOHAVEN THERAPEUTICS LTD.; BIOHAVEN PHARMACEUTICAL IRELAND DESIGNATED ACTIVITY COMPANY
Reel/Frame 071083/0330 →
PATENT SECURITY AGREEMENT Recorded Dec 2, 2021
From: BIOHAVEN THERAPEUTICS LTD.
To: SIXTH STREET SPECIALTY LENDING, INC., AS ADMINISTRATIVE AGENT
Reel/Frame 058299/0273 →
Continuity (3)
Provisional Application 62677018 · May 27, 2018
Provisional Application 62739774 · Oct 1, 2018
Related Publication 20220218673A1 · Jul 14, 2022
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