IP Library Granted Patent US 12,011,448
Granted Patent B2
US 12,011,448 · App. 17/056,931 · Granted Jun 18, 2024

Therapeutic or preventing agent for nephrotic syndrome including indole compound

Inventors: Yoshifumi Ueda (Takatsuki, JP); Takafumi Kurimoto (Takatsuki, JP)
Assignee: Japan Tobacco Inc.
A61K31/5377A61P13/12
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Quick Facts
Patent No.
US 12,011,448
App. No.
17/056,931
Granted
Jun 18, 2024
Kind
B2
Abstract

The present invention provides a therapeutic agent or prophylactic agent for nephrotic syndrome, containing N-[2-(6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1H-indol-6-yl]-N-methyl-(2S)-2-(morpholin-4-yl)propanamide or a pharmaceutically acceptable salt thereof.

Claims (10)

1. A method for treating nephrotic syndrome in a human subject in need thereof, comprising administering to the human subject a therapeutically effective amount of a compound represented by the following chemical structural formula:

or a pharmaceutically acceptable salt thereof.

2. The method according to claim 1 , wherein the nephrotic syndrome is primary nephrotic syndrome or secondary nephrotic syndrome.

3. The method according to claim 1 , wherein the nephrotic syndrome is at least one symptom of nephrotic syndrome selected from the group consisting of hypoalbuminemia, hypoproteinemia, dyslipidemia, immune disorder, edema and hypercholesterolemia.

4. The method according to claim 1 , wherein the pharmaceutically acceptable salt is monohydrochloride.

5. A method for preventing nephrotic syndrome in a human subject in need thereof, comprising administering to the human subject a therapeutically effective amount of a compound represented by the following chemical structural formula:

or a pharmaceutically acceptable salt thereof.

6. The method according to claim 5 , wherein the nephrotic syndrome is primary nephrotic syndrome or secondary nephrotic syndrome.

7. The method according to claim 5 , wherein the nephrotic syndrome is at least one symptom of nephrotic syndrome selected from the group consisting of hypoalbuminemia, hypoproteinemia, dyslipidemia, immune disorder, edema and hypercholesterolemia.

8. The method according to claim 5 , wherein the pharmaceutically acceptable salt is monohydrochloride.

Assignments (2)
NUNC PRO TUNC ASSIGNMENT Recorded Apr 8, 2026
From: JAPAN TOBACCO INC.
To: SHIONOGI & CO., LTD.
Reel/Frame 074312/0259 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 3, 2022
From: UEDA, YOSHIFUMI; KURIMOTO, TAKAFUMI
To: JAPAN TOBACCO INC.
Reel/Frame 059157/0453 →
Priority Claims (1)
JP 2018100669 · May 25, 2018 · national
Continuity (1)
Related Publication 20210236502A1 · Aug 5, 2021