IP Library Granted Patent US 12,458,646
Granted Patent B2
US 12,458,646 · App. 17/056,947 · Granted Nov 4, 2025

Therapeutic or preventing agent for multiple sclerosis including indole compound

Inventors: Yoshifumi Ueda (Takatsuki, JP); Takafumi Kurimoto (Takatsuki, JP); Naofumi Uesato (Takatsuki, JP)
Assignee: Japan Tobacco Inc.
A61K31/5377A61P25/28
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Quick Facts
Patent No.
US 12,458,646
App. No.
17/056,947
Granted
Nov 4, 2025
Kind
B2
Abstract

The present invention provides a therapeutic agent or prophylactic agent for multiple sclerosis, containing N-[2-(6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-3-yl)-1H-indol-6-yl]-N-methyl-(2S)-2-(morpholin-4-yl)propanamide or a pharmaceutically acceptable salt thereof.

Claims (8)

1 . A method for treating multiple sclerosis in a human subject in need thereof, comprising administering to the human subject a therapeutically effective amount of a compound represented by the following chemical structural formula:

or a pharmaceutically acceptable salt thereof, wherein the human subject has had a prior treatment with FTY-720, and wherein the prior treatment with FTY-720 is clinically insufficient.

2 . The method according to claim 1 , wherein the multiple sclerosis is selected from the group consisting of relapsing-remitting multiple sclerosis, primary progressive multiple sclerosis, and secondary progressive multiple sclerosis.

3 . The method according to claim 1 , wherein the human subject has at least one symptom of multiple sclerosis selected from the group consisting of feeling of weakness, ataxia, sensory neuropathy, dysuria, dyschezia, mental disorder and memory disorder.

4 . The method according to claim 1 , wherein the pharmaceutically acceptable salt is monohydrochloride.

5 . A method for suppressing the progression of a physical disorder of multiple sclerosis in a human subject in need thereof, comprising administering to the human subject a therapeutically effective amount of a compound represented by the following chemical structural formula:

or a pharmaceutically acceptable salt thereof, wherein the human subject has had a prior treatment with FTY-720, and wherein the prior treatment with FTY-720 is clinically insufficient.

6 . The method according to claim 5 , wherein the pharmaceutically acceptable salt is monohydrochloride.

Assignments (2)
NUNC PRO TUNC ASSIGNMENT Recorded Apr 8, 2026
From: JAPAN TOBACCO INC.
To: SHIONOGI & CO., LTD.
Reel/Frame 074312/0259 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 3, 2022
From: UEDA, YOSHIFUMI; KURIMOTO, TAKAFUMI; UESATO, NAOFUMI
To: JAPAN TOBACCO INC.
Reel/Frame 059311/0868 →
Priority Claims (1)
JP 2018-100668 · May 25, 2018 · national
Continuity (1)
Related Publication 20210236503A1 · Aug 5, 2021
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