IP Library Granted Patent US 11,357,844
Granted Patent B2
US 11,357,844 · App. 17/061,891 · Granted Jun 14, 2022

Isolated polypeptide of the toxin A and toxin B proteins of

Inventors: Larry R. Ellingsworth (Rockville, MD); David Flyer (Olney, MD); Jing-Hui Tian (Germantown, MD); Steven R. Fuhrmann (Germantown, MD); Stefanie Kluepfel-Stahl (Bethesda, MD); Gregory M. Glenn (Gaithersburg, MD); Kerstin Westritschnig (Vienna, AT)
Assignees: Valneva Austria GmbH; Valneva USA, Inc.
A61K39/08C07K14/33C07K16/1282A61K2039/53A61K2039/55505A61K2039/55544A61K2039/575C07K2317/76C07K2319/00C07K2319/40C07K2319/55
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Quick Facts
Patent No.
US 11,357,844
App. No.
17/061,891
Granted
Jun 14, 2022
Kind
B2
Abstract

This present invention provides C-TAB.G5 and C-TAB.G5.1 isolated polypeptides comprising the receptor binding domains of C. difficile toxin A and toxin B as set forth in the amino acid sequences of SEQ ID NO: 2 and SEQ ID NO: 4. The C-TAB.G5 and C-TAB.G5.1 isolated polypeptides may be used to neutralize toxic effects of C. difficile toxin A and/or toxin B.

Claims (25)

1. A method for producing a recombinant polypeptide derived from Clostridium difficile toxins A and B, the method comprising

i) introducing a recombinant nucleic acid encoding said polypeptide into a host cell, and

ii) culturing the host cell under conditions that allow expression of said polypeptide, wherein the polypeptide comprises an amino acid sequence having at least 85% sequence identity to the amino acid sequence as set forth in SEQ ID NO: 4, wherein the sequence identity is determined by Needleman-Wunsch global alignment.

2. The method of claim 1 , wherein the polypeptide comprises 19 repeating units of the C-terminal domain of toxin A.

3. The method of claim 1 , wherein the polypeptide comprises at least 23 repeating units of the C-terminal domain of toxin B.

4. The method of claim 1 , wherein the polypeptide has the amino acid sequence of SEQ ID NO: 2 or SEQ ID NO: 4.

5. The method of claim 1 , wherein the polypeptide is capable of inducing neutralizing antibodies against both C. difficile toxins A and B.

6. The method of claim 1 , wherein the polypeptide is useful for the treatment and/or prevention of C. difficile associated disease (CDAD) or infection.

7. The method for producing the polypeptide of claim 1 , wherein the method further comprises

iii) isolating said polypeptide.

8. The method of claim 1 , wherein the host cell is E. coli.

9. A method for producing a pharmaceutical composition comprising a recombinant polypeptide derived from Clostridium difficile toxins A and B, the method comprising combining the recombinant polypeptide and a pharmaceutically acceptable carrier or excipient, wherein the polypeptide comprises an amino acid sequence having at least 85% sequence identity to the amino acid sequence as set forth in SEQ ID NO: 4, wherein the sequence identity is determined by Needleman-Wunsch global alignment.

10. The method of claim 9 , wherein the polypeptide comprises 19 repeating units derived from the C-terminal domain of toxin A of C. difficile.

11. The method of claim 9 , wherein the polypeptide comprises at least 23 repeating units of the C-terminal domain of toxin B of C. difficile.

12. The method of claim 9 , wherein the polypeptide comprises the amino acid sequence of SEQ ID NO: 2 or SEQ ID NO: 4.

13. The method of claim 9 , wherein the composition is capable of inducing neutralizing antibodies against C. difficile toxins A and B.

14. A nucleic acid comprising a nucleic acid sequence encoding a polypeptide comprising an amino acid sequence having at least 85% sequence identity to the amino acid sequence as set forth in SEQ ID NO: 2 or SEQ ID NO: 4, wherein the sequence identity is determined by Needleman-Wunsch global alignment.

15. The nucleic acid of claim 14 , wherein the nucleic acid sequence encodes a polypeptide comprising an amino acid sequence having at least 95% sequence identity to the amino acid sequence as set forth in SEQ ID NO: 2 or SEQ ID NO: 4.

16. The nucleic acid of claim 14 , wherein the nucleic acid sequence encodes a polypeptide comprising the amino acid sequence having at least 99% sequence identity to the amino acid sequence as set forth in SEQ ID NO: 2 or SEQ ID NO: 4.

17. The nucleic acid of claim 14 , wherein the polypeptide comprises 19 repeating units derived from the C-terminal domain of toxin A of C. difficile and/or at least 23 repeating units of the C-terminal domain of toxin B of C. difficile.

18. The nucleic acid of claim 14 , wherein the nucleic acid sequence encodes a polypeptide consisting of the amino acid sequence as set forth in SEQ ID NO: 2.

19. The nucleic acid of claim 14 , wherein the nucleic acid sequence encodes a polypeptide consisting of the amino acid sequence as set forth in SEQ ID NO: 4.

20. A method for producing the nucleic acid of claim 14 , the method comprising:

i) amplifying a nucleic acid comprising the nucleic acid sequence; and/or

ii) introducing a vector comprising the nucleic acid sequence into a host cell, culturing the host cell under conditions that allow replication of the vector, and isolating the vector.

Assignments (6)
RELEASE OF SECURITY INTEREST Recorded Nov 10, 2025
From: WILMINGTON TRUST, NATIONAL ASSOCIATION, AS ADMINISTRATIVE AGENT
To: VALNEVA AUSTRIA GMBH; VALNEVA SE; VALNEVA USA, INC.
Reel/Frame 073516/0522 →
PATENT SECURITY AGREEMENT Recorded Oct 20, 2025
From: VALNEVA AUSTRIA GMBH; VALNEVA SE; VALNEVA SWEDEN AB
To: BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT
Reel/Frame 073164/0032 →
SECURITY INTEREST Recorded Jan 19, 2024
From: VALNEVA SE; VALNEVA AUSTRIA GMBH; VALNEVA USA, INC.; VALNEVA SWEDEN AB
To: WILMINGTON TRUST, NATIONAL ASSOCIATION
Reel/Frame 066182/0174 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 9, 2022
From: ELLINGSWORTH, LARRY R.; FLYER, DAVID; TIAN, JING-HUI; FUHRMANN, STEVEN R.; KLUEPFEL-STAHL, STEFANIE; GLENN, GREGORY M.
To: INTERCELL USA, INC.
Reel/Frame 059866/0717 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 9, 2022
From: WESTRITSCHNIG, KERSTIN
To: VALNEVA AUSTRIA GMBH
Reel/Frame 059912/0047 →
CHANGE OF NAME Recorded May 9, 2022
From: INTERCELL USA, INC.
To: VALNEVA USA, INC.
Reel/Frame 059912/0050 →