IP Library Granted Patent US 11,111,262
Granted Patent B2
US 11,111,262 · App. 17/063,947 · Granted Sep 7, 2021

C-mannoside compounds useful for the treatment of urinary tract infections

Inventors: Michael Joseph Bishop (Research Triangle Park, NC); Eugene L. Stewart (Collegeville, PA); Katherine Louisa Widdowson (San Diego, CA); James Walter Janetka (St. Louis, MO); Laurel Kathryn McGrane (St. Louis, MO)
Assignees: GlaxoSmithKline Intellectual Property Development Limited; Fimbrion Therapeutics, Inc.
C07H7/04A61K9/0014A61K9/0053A61K9/20A61K9/48A61K45/06
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Quick Facts
Patent No.
US 11,111,262
App. No.
17/063,947
Granted
Sep 7, 2021
Kind
B2
Abstract

Disclosed herein are new C-mannoside compounds and compositions and their application as pharmaceuticals for the treatment of human disease. Methods of inhibition of FimH activity in a human subject are also provided for the treatment diseases such as urinary tract infection.

Claims (4)

1. A compound which is

2. A pharmaceutical composition comprising the compound as recited in claim 1 together with a pharmaceutically acceptable carrier.

3. A pharmaceutical composition as recited in claim 2 formulated for oral administration.

4. The pharmaceutical composition as recited in claim 3 , wherein said composition is chosen from a tablet and a capsule.

Assignments (3)
CHANGE OF ADDRESS Recorded Oct 8, 2025
From: GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
Reel/Frame 073032/0390 →
CHANGE OF ADDRESS Recorded Jun 17, 2025
From: GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED
Reel/Frame 071649/0432 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 6, 2020
From: BISHOP, MICHAEL JOSEPH; STEWART, EUGENE L.; COLANDREA, VINCENT J.; STRAMBEANU, IULIA; LI, YUEHU; WIDDOWSON, KATHERINE LOUISA; MCGRANE, LAUREL KATHRYN; JANETKA, JAMES WALTER
To: GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED; FIMBRION THERAPEUTICS, INC.
Reel/Frame 053986/0701 →
Continuity (4)
Continuation PCTIB2019055806 · Jul 8, 2019
Provisional Application 62695993 · Jul 10, 2018
Provisional Application 62755588 · Nov 5, 2018
Related Publication 20210017212A1 · Jan 21, 2021
Cited By (1)
US 12,297,223