IP Library Granted Patent US 11,077,079
Granted Patent B1
US 11,077,079 · App. 17/118,041 · Granted Aug 3, 2021

GHB formulation and method for its manufacture

Inventors: Clark Allphin (Seattle, WA); Scott Bura (Gilroy, CA)
Assignee: Jazz Pharmaceuticals Ireland Limited
A61K31/19A61K9/5031A61K31/785A61K38/02
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 11,077,079
App. No.
17/118,041
Granted
Aug 3, 2021
Kind
B1
Abstract

The present application relates to GHB formulations and methods for manufacturing the same.

Claims (26)

1. A method of treating narcolepsy in a patient in need thereof, the method comprising:

administering a single daily dose to the patient, the single daily dose comprising an amount of oxybate equivalent to from 4.0 g to 12.0 g of sodium oxybate, wherein the administering comprises:

opening a sachet containing a solid oxybate formulation,

mixing the formulation with water, and

orally administering the mixture to the patient, wherein the oxybate formulation comprises an immediate release component and a controlled release component.

2. The method of claim 1 , wherein the orally administering occurs at night.

3. The method of claim 1 , wherein the oxybate formulation is mixed with water immediately prior to administration.

4. The method of claim 1 , wherein the oxybate is administered with food.

5. The method of claim 1 , wherein the administering promotes the patient to sleep for 6 to 8 hours.

6. The method of claim 1 , wherein the amount of oxybate administered to the patient is 35 mEq, 45 mEq, 60 mEq, or 70 mEq of oxybate.

7. The method of claim 1 , wherein the mixture is a suspension.

8. The method of claim 1 , wherein the oxybate formulation further comprises an acid.

9. The method of claim 8 , wherein the acid is selected from the group consisting of malic acid, citric acid, tartaric acid, boric acid, maleic acid, phosphoric acid, and benzoic acid.

10. A method of treating cataplexy or excessive daytime sleepiness associated with narcolepsy in a patient in need thereof, the method comprising:

administering a single daily dose to the patient, the single daily dose comprising an amount of oxybate equivalent to from 4.0 g to 12.0 g of sodium oxybate, wherein the administering comprises:

opening a sachet containing a solid oxybate formulation,

mixing the formulation with water, and

orally administering the mixture to the patient, wherein the oxybate formulation comprises an immediate release component and a controlled release component.

11. The method of claim 10 , wherein the orally administering occurs at night.

12. The method of claim 10 , wherein the oxybate formulation is mixed with water immediately prior to administration.

13. The method of claim 10 , wherein the oxybate is administered with food.

14. The method of claim 10 , wherein the administering promotes the patient to sleep for 6 to 8 hours.

15. The method of claim 10 , wherein the amount of oxybate administered to the patient is 35 mEq, 45 mEq, 60 mEq, or 70 mEq of oxybate.

16. The method of claim 10 , wherein the mixture is a suspension.

17. The method of claim 16 , wherein the oxybate formulation further comprises an acid.

18. The method of claim 17 , wherein the acid is selected from the group consisting of malic acid, citric acid, tartaric acid, boric acid, maleic acid, phosphoric acid, and benzoic acid.

Assignments (3)
SECURITY AGREEMENT Recorded May 5, 2021
From: CAVION, INC.; CELATOR PHARMACEUTICALS, INC.; JAZZ PHARMACEUTICALS IRELAND LIMITED; JAZZ PHARMACEUTICALS, INC.
To: U.S. BANK NATIONAL ASSOCIATION
Reel/Frame 056151/0010 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 15, 2020
From: JAZZ PHARMACEUTICALS, INC.
To: JAZZ PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 054649/0603 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Dec 14, 2020
From: ALLPHIN, CLARK; BURA, SCOTT
To: JAZZ PHARMACEUTICALS, INC.
Reel/Frame 054631/0826 →
Cited By (16)
US 12,226,377 US 12,226,388 US 12,226,389 US 12,239,625 US 12,257,223 US 12,263,150 US 12,263,151 US 12,295,926 US 12,303,478 US 12,337,066 US 12,396,956 US 12,440,449 US 12,478,604 US 12,551,457 US 12,582,622 US 12,691,090