IP Library Granted Patent US 11,141,457
Granted Patent B1
US 11,141,457 · App. 17/135,328 · Granted Oct 12, 2021

Oral octreotide therapy and contraceptive methods

Inventors: Asi Haviv (Gan-Shlomo, IL); Ruth Engle Stevens (Long Beach, WA); Jennings Ray Dawkins (Coats, NC)
Assignee: AMRYT ENDO, INC.
A61K38/12A61K9/0053
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Quick Facts
Patent No.
US 11,141,457
App. No.
17/135,328
Granted
Oct 12, 2021
Kind
B1
Abstract

This invention relates to methods of administering oral octreotide therapy to a female subject relating to avoidance of combined oral contraceptives or use of a back-up method for contraception.

Claims (18)

1. A method of administering oral octreotide to a female subject in need thereof wherein said subject is also in need of a contraceptive method, comprising

(a) administering to the subject oral octreotide; and

(b) counseling the subject to avoid concomitant use of a combined oral contraceptive.

2. The method of claim 1 , wherein the combined oral contraceptive comprises levonorgestrel.

3. A method of administering oral octreotide to a female subject in need thereof wherein said subject is administered a combined oral contraceptive, comprising

(a) administering to the subject oral octreotide; and

(b) counseling the subject to use a back-up method of contraception or to use an alternative non-hormonal method of contraception.

4. The method of claim 3 , wherein the combined oral contraceptive comprises levonorgestrel.

5. The method of claim 1 , wherein the subject has acromegaly.

6. The method of claim 1 , wherein the subject has severe diarrhea or flushing episodes associated with metastatic carcinoid tumor.

7. The method of claim 3 , wherein the subject has acromegaly.

8. The method of claim 3 , wherein the subject has severe diarrhea or flushing episodes associated with metastatic carcinoid tumor.

9. A method of administering oral octreotide to a female subject in need thereof wherein said subject is also in need of a contraceptive method, comprising

(a) administering to the subject oral octreotide; and

(b) counseling the subject to avoid concomitant use of a contraceptive which comprises levonorgestrel or to use a back-up method of contraception or to use an alternative method of contraception.

10. The method of claim 9 , wherein the contraceptive which comprises levonorgestrel is an oral contraceptive.

11. The method of claim 9 , wherein the contraceptive which comprises levonorgestrel is not an oral contraceptive.

12. The method of claim 11 , wherein the contraceptive is an intrauterine device.

Assignments (6)
MERGER AND CHANGE OF NAME Recorded Jan 7, 2026
From: AMRYT ENDO, INC.; AMYRT PHARMACEUTICALS INC.
To: AMRYT PHARMACEUTICALS INC.
Reel/Frame 073389/0551 →
CHANGE OF ADDRESS Recorded Mar 19, 2024
From: MCEVOY, JOHN
To: AMRYT ENDO, INC.
Reel/Frame 066833/0786 →
RELEASE OF SECURITY INTEREST Recorded Apr 13, 2023
From: ARES CAPITAL CORPORATION, AS ADMINISTRATIVE AGENT
To: AMRYT GENETICS LIMITED; AMRYT PHARMACEUTICALS, INC.; AMRYT ENDO, INC.; AMRYT RESEARCH LIMITED
Reel/Frame 063318/0849 →
SECURITY INTEREST Recorded Feb 18, 2022
From: AMRYT ENDO, INC.
To: ARES CAPITAL CORPORATION, AS ADMINISTRATIVE AGENT
Reel/Frame 059048/0944 →
MERGER Recorded Sep 7, 2021
From: CHIASMA, INC.
To: AMRYT ENDO, INC.
Reel/Frame 057401/0729 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 22, 2021
From: HAVIV, ASI; STEVENS, RUTH ENGLE; DAWKINS, JENNINGS RAY
To: CHIASMA, INC.
Reel/Frame 054994/0506 →