IP Library Granted Patent US 12,642,271
Granted Patent B2
US 12,642,271 · App. 17/164,293 · Granted Jun 2, 2026

Active compound combinations comprising a (thio)carboxamide derivative and a fungicidal compound

Inventors: Peter Dahmen (Neuss, DE); Philippe Desbordes (Lyons, FR); Christophe Dubost (Charbonnieres-les-Bains, FR); Stéphanie Gary (Champagne-au-Mont-d'Or, FR); Frank Goehlich (Hilden, DE); Hendrik Helmke (Liederbach, DE); Thomas Seitz (Langenfeld, DE); Ulrike Wachendorff-Neumann (Neuwied, DE); Ingo Wetcholowsky (Langenfeld, DE)
Assignee: Bayer CropScience Aktiengesellschaft
A01N43/56A01N43/40A01N43/50A01N43/54A01N43/653A01N43/84A01N55/00A01N59/20
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Quick Facts
Patent No.
US 12,642,271
App. No.
17/164,293
Granted
Jun 2, 2026
Kind
B2
Abstract

The present invention relates to active compound combinations, in particular within a fungicide composition, which comprises (A) a N-cyclopropyl-N-[substituted-benzyl]-3-(difluoromethyl)-5-fluoro-1-methyl-1H-pyrazole-4-carboxamide or thiocarboxamide derivative and a further fungicidally active compound (B). Moreover, the invention relates to a method for curatively or preventively or eradicatively controlling the phytopathogenic fungi of plants or crops, to the use of a combination according to the invention for the treatment of seed, to a method for protecting a seed and not at least to the treated seed.

Claims (20)

1 . A fungicidal composition comprising:

(A) a compound of formula (I):

wherein T represents an oxygen atom and X is 5-chloro-2-isopropyl; and

(B1) at least one further active fungicidal compound selected from the group consisting of: cyproconazole, epoxiconazole, fenhexamid, metconazole, propiconazole, prothioconazole, spiroxamine, tebuconazole, difenoconazole, bixafen, fluopyram, isopyrazam species selected from the group consisting of a mixture of syn-epimeric racemate 1RS,4SR,9RS and anti-epimeric racemate 1RS,4SR,9SR, syn-epimeric racemate 1RS,4SR,9RS, syn-epimeric enantiomer 1R,4S,9R, syn-epimeric enantiomer 1S,4R,9S, anti-epimeric racemate 1RS,4SR,9SR, anti-epimeric enantiomer 1R,4S,9S, and anti-epimeric enantiomer 1S,4R,9R; penflufen, penthiopyrad, sedaxane, fluxapyroxad, benzovindiflupyr, azoxystrobin, fluoxastrobin, pyraclostrobin, trifloxystrobin, folpet, pyrimethanil, metalaxyl, fludioxonil, and (3S,6S,7R,8R)-8-benzyl-3-[({3-[(isobutyryloxy)methoxy]-4-methoxypyridin-2-yl}carbonyl)amino]-6-methyl-4,9-dioxo-1,5-dioxonan-7-yl-2-methylpropanoate,

wherein each of (A) and (B1) is present in the composition at active but non-phytotoxic amounts, and

wherein the weight ratio of (A):(B1) is in a range of 1:1 to 1:20, the concentration of (A) is 0.125 to 40 ppm, the concentration of (B1) is 0.125 to 400 ppm, and the composition results in a synergistic fungicidal effect.

2 . The composition according to claim 1 , comprising at least one further active ingredient selected from the group consisting of insecticides, attractants, sterilants, bactericides, acaricides, nematicides, fungicides, growth regulators, herbicides, fertilizers, safeners and semiochemicals.

3 . The composition according to claim 1 , wherein the isopyrazam species a mixture of syn-epimeric racemate 1RS,4SR,9RS and anti-epimeric racemate 1RS,4SR,9SR.

4 . The composition according to claim 1 , wherein the weight ratio of (A):(B1) is in a range of 1:1 to 1:10.

5 . The composition according to claim 1 , wherein (B1) is selected from the group consisting of fenhexamid, prothioconazole, tebuconazole, difenoconazole, fluopyram, pyraclostrobin, trifloxystrobin, and (3S,6S,7R,8R)-8-benzyl-3-[({3-[(isobutyryloxy)methoxy]-4-methoxypyridin-2-yl}carbonyl)amino]-6-methyl-4,9-dioxo-1,5-dioxonan-7-yl-2-methylpropanoate.

6 . The composition according to claim 1 , wherein (B1) is fluopyram, and wherein the weight ratio of (A):(B1) is in a range of 1:1 to 1:10.

7 . A composition for controlling phytopathogenic harmful fungi, comprising a composition according to claim 1 , in addition to extenders and/or surfactants.

8 . A method for controlling phytopathogenic harmful fungi, comprising applying a composition according to claim 1 to the phytopathogenic harmful fungi and/or their habitat.

9 . The method according to claim 8 , wherein the phytopathogenic harmful fungi is of the Phytophthora, Venturia, Alternaria, Sphaerotheca, Botrytis, Blumeria, Fusarium, Leptosphaeria, Puccinia, Pyrenophora , or Septoria species.

10 . A process for producing compositions for controlling phytopathogenic harmful fungi, comprising mixing a composition according to claim 1 with extenders and/or surfactants.

11 . The method according to claim 10 , wherein the phytopathogenic harmful fungi is of the Phytophthora, Venturia, Alternaria, Sphaerotheca, Botrytis, Blumeria, Fusarium, Leptosphaeria, Puccinia, Pyrenophora , or Septoria species.

12 . A method for the treatment of transgenic plants, comprising applying a composition according to claim 1 to said transgenic plants.

13 . The method according to claim 12 , wherein the transgenic plant is tomato, apple, cucumber, bean, barley, or wheat.

14 . A method for the treatment of seed or of seed of transgenic plants, comprising applying a composition according to claim 1 to said seed or to said transgenic plants.

15 . The method according to claim 14 , wherein the transgenic plant is tomato, apple, cucumber, bean, barley, or wheat.

Assignments (4)
NUNC PRO TUNC ASSIGNMENT Recorded Jul 4, 2023
From: BAYER INTELLECTUAL PROPERTY GMBH
To: BAYER CROPSCIENCE AKTIENGESELLSCHAFT
Reel/Frame 064198/0823 →
CHANGE OF ADDRESS Recorded Jun 12, 2023
From: BAYER INTELLECTUAL PROPERTY GMBH
To: BAYER INTELLECTUAL PROPERTY GMBH
Reel/Frame 064021/0344 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 14, 2021
From: DAHMEN, PETER; DESBORDES, PHILIPPE; DUBOST, CHRISTOPHE; GARY, STEPHANIE; GOEHLICH, FRANK; HELMKE, HENDRIK; SEITZ, THOMAS; WACHENDORFF-NEUMANN, ULRIKE; WETCHOLOWSKY, INGO
To: BAYER INTELLECTUAL PROPERTY GMBH
Reel/Frame 055920/0354 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 14, 2021
From: BAYER INTELLECTUAL PROPERTY GMBH
To: BAYER CROPSCIENCE AKTIENGESELLSCHAFT
Reel/Frame 055920/0362 →
Priority Claims (1)
EP 11356005 · Apr 22, 2011 · regional
Continuity (3)
Division 14112375
Provisional Application 61486479 · May 16, 2011
Related Publication 20210227828A1 · Jul 29, 2021
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