IP Library Granted Patent US 11,492,412
Granted Patent B2
US 11,492,412 · App. 17/190,792 · Granted Nov 8, 2022

Preparations and methods for treating a GD2 positive cancer

Inventors: Hans Loibner (Vienna, AT); Oliver Mutschlechner (Wiener Neudorf, AT); Ruth Ladenstein (Vienna, AT); Isabel Klier (Vienna, AT)
Assignee: APEIRON BIOLOGICS AG
C07K16/3084A61K9/0019A61K2039/505A61K2039/545C07K2317/24C07K2317/734
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Quick Facts
Patent No.
US 11,492,412
App. No.
17/190,792
Granted
Nov 8, 2022
Kind
B2
Abstract

A method of treating a high-risk neuroblastoma in a patient is described.

Claims (45)

1. A method of treating a high-risk neuroblastoma in a patient, the method comprising:

administering to the patient a ch14.18/CHO chimeric anti-GD2 antibody or a ch14.18/SP2/0 chimeric anti-GD2 antibody at a dose of 17.5 mg/m 2 /day over at least 10 hours per day over 4 consecutive days in a cycle having from 24 to 32 days;

wherein

the administering of the anti-GD2 antibody is for a total of 5 cycles;

in each of cycles 1, 3, and 5 of the 5 cycles, the administering of the anti-GD2 antibody is on the fourth day to the seventh day of each of the cycles 1, 3, and 5;

in each of cycles 2 and 4 of the 5 cycles, the administering of the anti-GD2 antibody is on the eighth day to the eleventh day of each of the cycles 2 and 4; and

administering retinoic acid in each of cycles 1, 3, and 5 of the 5 cycles on the eleventh day to the twenty-fourth day of the cycles 1, 3, and 5; and

administering retinoic acid in each of cycles 2 and 4 of the 5 cycles on the fifteenth day to the twenty-eighth day of the cycles 2 and 4.

2. The method of claim 1 , wherein the patient is a pediatric patient.

3. The method of claim 2 , wherein the retinoic acid is administered orally twice daily for a total dose of 160 mg/m 2 /day.

4. The method of claim 3 , further comprising in each of cycles 1, 3, and 5 of the 5 cycles, administering GM-CSF on the first day to the fourteenth day of the cycles 1, 3, and 5, wherein the GM-CSF is administered at a dose of 250 μg/m 2 /day by subcutaneous injection or by IV infusion over 2 hours.

5. The method of claim 4 , further comprising in each of cycles 2 and 4 of the 5 cycles, administering IL-2 on the first day to the fourth day and on the eighth day to the eleventh day of the cycles 2 and 4, wherein the IL-2 is administered at a dose of 3 MIU/m 2 /day by continuous IV infusion over 96 hours on the first day to the fourth day and at a dose of 4.5 MIU/m 2 /day on the eighth day to the eleventh day.

6. The method of claim 1 , wherein the anti-GD2 antibody is administered for at least 10 hours per day up to 20 hours per day.

7. The method of claim 1 , wherein the patient has previously been treated with one or more therapies selected from the group consisting of surgery, chemotherapy, radiation therapy, myeloablative therapy (MAT), metaiodobenzylguanidine scintigraphy (mIBG), vaccine therapy, stem cell transplantation, and retinoid treatment.

8. The method of claim 7 , wherein the stem cell transplantation is an autologous stem cell transplantation.

9. A method of treating a high-risk neuroblastoma in a patient, the method comprising:

administering to the patient a ch14.18/CHO chimeric anti-GD2 antibody or a ch14.18/SP2/0 chimeric anti-GD2 antibody at a dose of 17.5 mg/m 2 /day as an intravenous infusion over 4 consecutive days;

wherein the anti-GD2 antibody comprises a heavy chain and a light chain, the heavy chain encoded by the nucleic acid sequence of SEQ ID NO:2 and the light chain encoded by the nucleic acid sequence of SEQ ID NO:1;

wherein the patient has previously been treated with one or more therapies selected from the group consisting of surgery, chemotherapy, radiation therapy, myeloablative therapy (MAT), metaiodobenzylguanidine scintigraphy (mIBG), vaccine therapy, stem cell transplantation, and retinoid treatment.

10. The method of claim 9 , wherein the patient is a pediatric patient.

11. The method of claim 9 , wherein the stem cell transplantation is an autologous stem cell transplantation.

12. The method of claim 9 , wherein the 4 consecutive days are comprised in a cycle having from 24 to 32 days.

13. The method of claim 12 , wherein the administering is for one treatment period of 4 consecutive days per cycle, for a total of 5 cycles.

14. The method of claim 13 , wherein in each of cycles 1, 3, and 5 of the 5 cycles, the administering of the anti-GD2 antibody is on the fourth day to the seventh day of each of the cycles 1, 3, and 5, and in each of cycles 2 and 4 of the 5 cycles, the administering of the anti-GD2 antibody is on the eighth day to the eleventh day of each of the cycles 2 and 4.

15. The method of claim 14 , further comprising:

administering retinoic acid in each of cycles 1, 3, and 5 of the 5 cycles on the eleventh day to the twenty-fourth day of the cycles 1, 3, and 5; and

administering retinoic acid in each of cycles 2 and 4 of the 5 cycles on the fifteenth day to the twenty-eighth day of the cycles 2 and 4.

16. The method of claim 15 , further comprising in each of cycles 1, 3, and 5 of the 5 cycles, administering GM-CSF on the first day to the fourteenth day of the cycles 1, 3, and 5.

17. The method of claim 9 , wherein the intravenous infusion is over at least 10 hours per day.

18. The method of claim 9 , wherein the intravenous infusion is over 10 or more hours per day up to 20 hours per day.

19. A method of treating a high-risk neuroblastoma in a patient, the method comprising:

administering to the patient a ch14.18/CHO chimeric anti-GD2 antibody or a ch14.18/SP2/0 chimeric anti-GD2 antibody at a dose of 17.5 mg/m 2 /day as an intravenous infusion over 4 consecutive days;

wherein the anti-GD2 antibody comprises a heavy chain and a light chain, the heavy chain encoded by the nucleic acid sequence of SEQ ID NO:2 and the light chain encoded by the nucleic acid sequence of SEQ ID NO:1;

wherein the 4 consecutive days are comprised in a cycle having from 24 to 32 days;

wherein the administering is for one treatment period of 4 consecutive days per cycle, for a total of 5 cycles; and

wherein in each of cycles 1, 3, and 5 of the 5 cycles, the administering of the anti-GD2 antibody is on the fourth day to the seventh day of each of the cycles 1, 3, and 5, and in each of cycles 2 and 4 of the 5 cycles, the administering of the anti-GD2 antibody is on the eighth day to the eleventh day of each of the cycles 2 and 4.

20. The method of claim 19 , further comprising:

administering retinoic acid in each of cycles 1, 3, and 5 of the 5 cycles on the eleventh day to the twenty-fourth day of the cycles 1, 3, and 5; and

administering retinoic acid in each of cycles 2 and 4 of the 5 cycles on the fifteenth day to the twenty-eighth day of the cycles 2 and 4.

21. The method of claim 20 , further comprising in each of cycles 1, 3, and 5 of the 5 cycles, administering GM-CSF on the first day to the fourteenth day of the cycles 1, 3, and 5.

22. The method of claim 19 , wherein the intravenous infusion is over at least 10 hours per day.

23. The method of claim 19 , wherein the intravenous infusion is over 10 or more hours per day up to 20 hours per day.

24. The method of claim 19 , wherein the patient is a pediatric patient.

25. The method of claim 19 , wherein the patient has previously been treated with one or more therapies selected from the group consisting of surgery, chemotherapy, radiation therapy, myeloablative therapy (MAT), metaiodobenzylguanidine scintigraphy (mIBG), vaccine therapy, stem cell transplantation, and retinoid treatment.

26. The method of claim 25 , wherein the stem cell transplantation is an autologous stem cell transplantation.

Assignments (3)
CHANGE OF NAME Recorded Jan 9, 2025
From: APEIRON BIOLOGICS AG
To: APEIRON BIOLOGICS GMBH
Reel/Frame 069856/0952 →
SECURITY INTEREST Recorded Dec 23, 2024
From: APEIRON BIOLOGICS GMBH
To: CITIBANK, N.A., AS ADMINISTRATIVE AGENT
Reel/Frame 069669/0908 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 15, 2022
From: LOIBNER, HANS; MUTSCHLECHNER, OLIVER; LADENSTEIN, RUTH; KLIER, ISABEL
To: APEIRON BIOLOGICS AG
Reel/Frame 059268/0102 →
Priority Claims (2)
CA CA 2834000 · Nov 21, 2013 · national
EP 13193953 · Nov 21, 2013 · regional
Continuity (6)
Continuation 16920880 · Jul 6, 2020
Continuation 15824055 · Nov 28, 2017
Continuation 15036519
Continuation In Part 14182776 · Feb 18, 2014
Continuation In Part 14086696 · Nov 21, 2013
Related Publication 20210221909A1 · Jul 22, 2021