IP Library Granted Patent US 12,220,414
Granted Patent B2
US 12,220,414 · App. 17/258,913 · Granted Feb 11, 2025

Use of sGC stimulators for the treatment of mitochondrial disorders

Inventor: John R. Hadcock (Cambridge, MA)
Assignee: Tisento Therapeutics Inc.
A61K31/506A61K31/197A61K31/401A61K31/5377A61P25/28
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Quick Facts
Patent No.
US 12,220,414
App. No.
17/258,913
Granted
Feb 11, 2025
Kind
B2
Abstract

The present disclosure relates to methods, uses, pharmaceutical compositions comprising an sGC stimulator or a pharmaceutically acceptable salt thereof, alone or in combination with one or more additional therapeutic agents, for the treatment of a mitochondrial disorder.

Claims (5)

1. A method of treating MELAS (Mitochondrial myopathy, encephalomyopathy, lactic acidosis, stroke-like symptoms) in a patient in need thereof, comprising administering to said patient a therapeutically effective amount of an sGC stimulator or a pharmaceutically acceptable salt thereof, wherein the sGC stimulator or a pharmaceutically acceptable salt thereof, is represented by the following formula:

or a pharmaceutically acceptable salt thereof.

2. The method of claim 1 , wherein said sGC stimulator, or a pharmaceutically acceptable salt thereof, is administered in combination with arginine or citrulline.

3. A method of treating MELAS (Mitochondrial myopathy, encephalomyopathy, lactic acidosis, stroke-like symptoms) in a patient in need thereof, comprising administering to said patient a therapeutically effective amount of an sGC stimulator, wherein the sGC stimulator is represented by the following formula:

4. The method of claim 3 , wherein said sGC stimulator is administered in combination with arginine or citrulline.

Assignments (3)
CORRECTIVE ASSIGNMENT TO CORRECT THE ASSIGNEE NAME FROM TISENTO THERAPEUTICS, INC. TO TISENTO THERAPEUTICS INC. PREVIOUSLY RECORDED ON REEL 064792 FRAME 0500. ASSIGNOR(S) HEREBY CONFIRMS THE ASSIGNMENT. Recorded Sep 13, 2023
From: CYCLERION THERAPEUTICS, INC.
To: TISENTO THERAPEUTICS INC.
Reel/Frame 064889/0459 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 1, 2023
From: CYCLERION THERAPEUTICS, INC.
To: TISENTO THERAPEUTICS, INC.
Reel/Frame 064792/0500 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 9, 2021
From: HADCOCK, JOHN R.
To: CYCLERION THERAPEUTICS, INC.
Reel/Frame 055198/0620 →
Continuity (3)
Provisional Application 62697671 · Jul 13, 2018
Provisional Application 62696582 · Jul 11, 2018
Related Publication 20210177846A1 · Jun 17, 2021
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