IP Library Granted Patent US 11,976,068
Granted Patent B2
US 11,976,068 · App. 17/357,008 · Granted May 7, 2024

7-benzyl-4-(2-methylbenzyl)-2,4,6,7,8,9-hexahydroimidazo [1,2-a]pyrido[3,4-e]pyrimidin-5(1H)-one, analogs thereof, and salts thereof and methods for their use in therapy

Inventors: Joshua E. Allen (New Haven, CT); Martin Stogniew (Lakewood Ranch, FL); Richard S. Pottorf (Indianapolis, IN); Bhaskara Rao Nallaganchu (Hillsborough, NJ); Gary Olson (Mountainside, NJ); Yanjun Sun (Kendall Park, NJ)
Assignee: ONCOCEUTICS, INC.
C07D471/14A61K31/337A61K31/519A61K45/06C07D471/12C07D487/14Y02A50/30
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Quick Facts
Patent No.
US 11,976,068
App. No.
17/357,008
Granted
May 7, 2024
Kind
B2
Abstract

This disclosure relates to methods of treatment using compound (1) or analogs thereof, and pharmaceutically acceptable salts thereof. Also disclosed are compounds of formula (10): as defined in the specification, and pharmaceutically acceptable salts thereof, as well as pharmaceutical compositions comprising the same. Methods of treatment, such as for cancer, are provided that comprise administering the compounds and their salts to a subject in need of such treatment.

Claims (6)

1. A pharmaceutical composition comprising:

a) a compound of formula (1)

or a pharmaceutically acceptable salt thereof in an amount of between about 100 mg to about 1000 mg, based on the free base weight; and

b) one or more pharmaceutically acceptable carrier,

wherein the pharmaceutically acceptable salt is a di-salt.

2. The composition of claim 1 , wherein the di-salt is a hydrochloride di-salt.

Assignments (4)
CONFIRMATORY PATENT ASSIGNMENT Recorded Oct 27, 2025
From: CHIMERIX, INC.; ONCOCEUTICS, INC.
To: JAZZ PHARMACEUTICALS IRELAND LIMITED
Reel/Frame 073333/0883 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2023
From: STOGNIEW, MARTIN; ALLEN, JOSHUA E.
To: ONCOCEUTICS, INC.
Reel/Frame 062706/0737 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2023
From: POTTORF, RICHARD S.; NALLAGANCHU, BHASKARA RAO; OLSON, GARY L.; SUN, YANJUN
To: PROVID PHARMACEUTICALS INC.
Reel/Frame 062706/0901 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2023
From: PROVID PHARMACEUTICALS INC.
To: ONCOCEUTICS, INC.
Reel/Frame 062760/0223 →