IP Library Granted Patent US 12,171,804
Granted Patent B2
US 12,171,804 · App. 17/374,302 · Granted Dec 24, 2024

Methods of treating chemotherapy induced neutropenia using fixed doses of eflapegrastim

Inventors: John A. Barrett (Groton, MA); Sribalaji Lakshmikanthan (Boxborough, MA)
Assignee: Spectrum Pharmaceuticals, Inc.
A61K38/193A61K45/06A61P7/06
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Quick Facts
Patent No.
US 12,171,804
App. No.
17/374,302
Granted
Dec 24, 2024
Kind
B2
Abstract

This disclosure provides a method of preventing, alleviating, or treating a condition (i.e., neutropenia) in a patient in need thereof, the condition characterized by compromised white blood cell production in the patient. The method includes administering to the patient a therapeutically effective amount of a protein complex comprising a modified human granulocyte-colony stimulating factor (hG-CSF) covalently linked to an immunoglobulin Fc region via a non-peptidyl polymer at a fixed dose regardless of the patient's weight.

Claims (9)

1. A method of preventing or reducing chemotherapy-induced neutropenia in a patient in need thereof wherein the patient is also being administered at least one cycle of a chemotherapy regimen, the method comprising administering to the patient a EFLAPEGRASTIM at a fixed dose of 13.2 mg regardless of patient's weight approximately 24 hours (±2 hours) after administration of the chemotherapy once per chemotherapy cycle wherein prior to administration of the EFLAPEGRASTIM, the patient exhibits an absolute neutrophil count of ≥1.5×10 9 /L and a platelet count ≥100×10 9 /L.

2. The method of claim 1 , wherein the neutropenia is severe chronic neutropenia or febrile neutropenia.

3. The method of claim 1 , wherein the chemotherapy regimen comprises at least one of docetaxel and cyclophosphamide.

4. The method of claim 1 , wherein the chemotherapy regimen comprises a combination of docetaxel and cyclophosphamide.

5. The method of claim 1 , wherein a second dose of the EFLAPEGRASTIM is administered between 5 and 30 days after a first dose of EFLAPEGRASTIM is administered to the patient.

6. The method of claim 5 , wherein the second dose of the EFLAPEGRASTIM is administered between 15 and 25 days after a first dose of EFLAPEGRASTIM is administered to the patient.

7. The method of claim 1 , wherein the patient's weight ranges from 30 kg to 180 kg.

8. The method of claim 1 , wherein the fixed dose is provided in a dosage volume of about 0.4 ml to about 1 ml.

9. The method of claim 8 , wherein the fixed dose is provided in a dosage volume of about 0.6 ml.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 1, 2026
From: SPECTRUM PHARMACEUTICALS, INC.
To: ASSERTIO SPECIALTY PHARMACEUTICALS, LLC
Reel/Frame 074542/0184 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 12, 2025
From: BARRETT, JOHN A.; LAKSHMIKANTHAN, SRIBALAJI
To: SPECTRUM PHARMACEUTICALS, INC.
Reel/Frame 072881/0226 →
TERMINATION AND RELEASE OF INTELLECTUAL PROPERTY SECURITY AGREEMENT RECORDED AT REEL 061179/FRAME 0202 Recorded Aug 1, 2023
From: SLR INVESTMENT CORP.
To: SPECTRUM PHARMACEUTICALS, INC.; ALLOS THERAPEUTICS, INC.; TALON THERAPEUTICS, INC.
Reel/Frame 064463/0709 →
SECURITY INTEREST Recorded Sep 22, 2022
From: SPECTRUM PHARMACEUTICALS, INC.; ALLOS THERAPEUTICS, INC.; TALON THERAPEUTICS, INC.
To: SLR INVESTMENT CORP., AS COLLATERAL AGENT
Reel/Frame 061179/0202 →