IP Library Granted Patent US 12,552,855
Granted Patent B2
US 12,552,855 · App. 17/608,743 · Granted Feb 17, 2026

CD33 targeted immunotherapies

Inventors: Jordan Jarjour (Cambridge, MA); Mark Pogson (Cambridge, MA); Wai-Hang Leung (Cambridge, MA); Kyle Jones (La Jolla, CA); William Crago (La Jolla, CA); Angelica Sanabria (La Jolla, CA); Andrew Hollands (La Jolla, CA); Jacob Gano (La Jolla, CA); Milton Ma (La Jolla, CA); John C. Timmer (La Jolla, CA); Brendan P. Eckelman (La Jolla, CA)
Assignees: Regeneron Pharmaceuticals, Inc.; Inhibrx Biosciences, Inc.
C07K14/70596A61K40/11A61K40/31A61K40/421A61P35/00C07K14/005C07K14/7051C07K14/70514C07K14/70517C07K14/70578C07K14/7151C07K16/2803C12N5/0636C12N9/90C12N15/86C12Y502/01008A61K38/00A61K2039/505A61K2239/38C07K2317/569C07K2317/622C07K2319/02C07K2319/03C07K2319/33C07K2319/50C07K2319/74C12N2740/15043C12N2740/15071
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Quick Facts
Patent No.
US 12,552,855
App. No.
17/608,743
Granted
Feb 17, 2026
Kind
B2
Abstract

The present disclosure provides improved CD33 targeting polypeptides and compositions for adoptive T cell therapies for treating, preventing, or ameliorating at least one symptom of a cancer, infectious disease, autoimmune disease, inflammatory disease, and immunodeficiency, or condition associated therewith.

Claims (26)

1 . A polypeptide complex comprising:

(a) a first polypeptide comprising:

(i) an FRB multimerization domain polypeptide;

(ii) a CD8α transmembrane domain or a CD4 transmembrane domain;

(iii) a CD137 co-stimulatory domain; and/or

(iv) a CD3ζ primary signaling domain; and

(b) a second polypeptide comprising:

(i) an anti-CD33 VHH antibody that has an amino acid sequence set forth in SEQ ID NO: 10;

(ii) an FKBP12 multimerization domain polypeptide; and

(iii) a CD4 transmembrane domain;

wherein the second polypeptide comprises the sequence set forth in SEQ ID NO: 30.

2 . The polypeptide complex of claim 1 , wherein the first polypeptide comprises the sequence set forth in SEQ ID NO: 82.

3 . The polypeptide complex of claim 1 , further comprising a bridging factor associated with and disposed between the multimerization domain polypeptides of the first and second polypeptides, wherein the bridging factor is selected from the group consisting of: AP21967, sirolimus, everolimus, novolimus, pimecrolimus, ridaforolimus, tacrolimus, temsirolimus, umirolimus, and zotarolimus.

4 . The polypeptide complex of claim 1 , wherein the second polypeptide comprises a costimulatory domain.

5 . The polypeptide complex of claim 4 , wherein the costimulatory domain of the second polypeptide is selected from a costimulatory molecule selected from the group consisting of: Toll-like receptor 1 (TLR1), TLR2, TLR3, TLR4, TLR5, TLR6, TLR7, TLR8, TLR9, TLR10, caspase recruitment domain family member 11 (CARD11), CD2, CD7, CD27, CD28, CD30, CD40, CD54 (ICAM), CD83, CD94, CD134 (OX40), CD137 (4-1BB), CD278 (ICOS), DNAX-Activation Protein 10 (DAP10), Linker for activation of T-cells family member 1 (LAT), SH2 domain-containing leukocyte protein of 76 kD (SLP76), T cell receptor associated transmembrane adaptor 1 (TRAT1), TNFR2, TNFRS14, TNFRS18, TNRFS25, and zeta chain of T cell receptor associated protein kinase 70 (ZAP70).

6 . The polypeptide complex of claim 4 , wherein the costimulatory domain of the second polypeptide is a costimulatory domain isolated from OX40 or TNFR2.

7 . The polypeptide complex of claim 1 , wherein the FRB multimerization domain polypeptide and the FKBP multimerization domain polypeptide localize extracellularly when of the first polypeptide and the second polypeptide are expressed.

8 . The polypeptide complex of claim 1 , wherein the polypeptide complex forms on the surface of a cell.

9 . The polypeptide complex of claim 8 , wherein the cell is:

a) a hematopoietic cell;

b) a T cell, an αβ T cell, or a γδ T cell;

c) a CD3+, CD4+, and/or CD8+ cell;

d) an immune effector cell;

e) a cytotoxic T lymphocytes (CTLs), a tumor infiltrating lymphocytes (TILs), or a helper T cell; and/or

f) a natural killer (NK) cell or natural killer T (NKT) cell;

wherein the source of the cell is peripheral blood mononuclear cells, bone marrow, lymph nodes tissue, cord blood, thymus issue, tissue from a site of infection, ascites, pleural effusion, spleen tissue, or tumors.

Assignments (7)
SECURITY INTEREST Recorded Jan 14, 2025
From: INHIBRX BIOSCIENCES, INC.
To: OXFORD FINANCE LLC; OXFORD FINANCE LLC
Reel/Frame 069894/0045 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 10, 2024
From: INHIBRX, INC.
To: INHIBRX BIOSCIENCES, INC.
Reel/Frame 067679/0338 →
RELEASE OF SECURITY INTEREST Recorded Jun 3, 2024
From: OXFORD FINANCE LLC, AS COLLATERAL AGENT
To: INHIBRX, INC.
Reel/Frame 067606/0247 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 22, 2024
From: 2SEVENTY BIO, INC.
To: REGENERON PHARMACEUTICALS, INC.
Reel/Frame 067184/0147 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 1, 2022
From: JONES, KYLE; CRAGO, WILLIAM; SANABRIA, ANGELICA; HOLLANDS, ANDREW; GANO, JACOB; MA, MILTON; TIMMER, JOHN C.; ECKELMAN, BRENDAN P.
To: INHIBRX, INC.
Reel/Frame 060970/0188 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 7, 2022
From: JARJOUR, JORDAN; POGSON, MARK; LEUNG, WAI-HANG
To: 2SEVENTY BIO, INC.
Reel/Frame 059181/0749 →
INTELLECTUAL PROPERTY SECURITY AGREEMENT Recorded Feb 28, 2022
From: INHIBRX, INC.
To: OXFORD FINANCE LLC
Reel/Frame 059262/0780 →
Continuity (3)
Provisional Application 62898392 · Sep 10, 2019
Provisional Application 62845304 · May 8, 2019
Related Publication 20220324942A1 · Oct 13, 2022
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