IP Library Granted Patent US 12,584,179
Granted Patent B2
US 12,584,179 · App. 18/130,547 · Granted Mar 24, 2026

DNA methylation and mutational analysis methods for bladder cancer surveillance

Inventors: Margarita Lopatin (Palo Alto, CA); Athanasios Tsiatis (San Francisco, CA); Christopher N. Silk (Redwood City, CA); David P. Miller (Albany, CA); Michael R. Crager (Menlo Park, CA); Phillip Febbo (Mill Valley, CA); Dejan Knezevic (Redwood City, CA)
Assignee: Genomic Health, Inc.
C12Q1/6886A61P35/00C12Q2600/106C12Q2600/154G01N2800/52G01N2800/56G01N2800/7028
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Quick Facts
Patent No.
US 12,584,179
App. No.
18/130,547
Granted
Mar 24, 2026
Kind
B2
Abstract

The present disclosure relates to methods of monitoring bladder cancer patients and analyzing patient samples for presence of methylated DNA and optionally particular gene mutations. In some embodiments, analysis results are correlated with clinical outcome measures such as risk of bladder cancer recurrence.

Claims (30)

1 . A method of characterizing a urine sediment sample obtained from a subject, comprising:

bisulfite converting DNA from the sample; and

performing methylation-specific quantitative PCR on the bisulfite converted DNA to determine the amount and/or the concentration of methylated DNA in the sample from a set of genes consisting of at least four genes selected from MEIS1, NKPD1, ONECUT2, KLF2, OSR1, SOX1, EOMES, DDX25, TMEM106A, EPHX3, IRX5, NID2, VIM, and ITPKB, wherein the set of genes comprises one or both of NKPD1 and KLF2, and from a set of one or more reference genes, wherein the reference gene(s) have a methylation level that is not significantly different in a subject with bladder cancer compared to a subject without bladder cancer.

2 . The method of claim 1 , wherein the subject has or is suspected of having bladder cancer.

3 . The method of claim 2 , wherein the subject has been diagnosed with non-muscle-invasive bladder cancer.

4 . The method of claim 2 , wherein the sample is obtained from the subject prior to cystoscopy or after a negative cystoscopy.

5 . The method of claim 1 , wherein the set of genes comprises both of NKPD1 and KLF2.

6 . The method of claim 1 , wherein the set of one or more reference genes comprises one or more of CTNS, TOP3A, COL2A and SLC24A3.

7 . The method of claim 1 , wherein the set of genes consists of one of the following gene sets:

(a) MEIS1, NKPD1, ONECUT2, KLF2;

(b) MEIS1, NKPD1, ONECUT2, OSR1;

(c) MEIS1, NKPD1, KLF2, SOX1;

(d) MEIS1, NKPD1, ONECUT2, OSR1, TMEM106A; EPHX3;

(e) MEIS1, NKPD1, ONECUT2, KLF2, TMEM106A, IRX5;

(f) MEIS1, NKPD1, ONECUT2, KLF2, SOX1, TMEM106A; or

(g) MEIS1, NKPD1, ONECUT2, KLF2, TMEM106A, ITPKB.

8 . The method of claim 1 , wherein the method further comprises analyzing the bisulfite converted DNA for mutations in one or both of FGFR3 and TERT.

9 . The method of claim 1 , wherein the set of genes consists of four genes wherein the four genes comprise MEIS1, NKPF1, and KLF2.

10 . A method of characterizing a urine sediment sample obtained from a subject, comprising:

bisulfite converting DNA from the sample; and

performing methylation-specific quantitative PCR on the bisulfite converted DNA to determine the amount and/or the concentration of methylated DNA in the sample from a set of genes consisting of three or four genes, wherein the set of three or four genes comprises one or both of NKPD1 and KLF2; and from a set of one or more reference genes wherein the reference gene(s) have a methylation level that is not significantly different in a subject with bladder cancer compared to a subject without bladder cancer.

11 . The method of claim 10 , wherein the subject has or is suspected of having bladder cancer.

12 . The method of claim 11 , wherein the subject has been diagnosed with non-muscle-invasive bladder cancer.

13 . The method of claim 11 , wherein the sample is obtained from the patient prior to cystoscopy or after a negative cystoscopy.

14 . The method of claim 10 , wherein the set of three or four genes consists of (a) one or both of NKPD1 and KLF2 and (b) one, two, or three genes selected from MEIS1, ONECUT2, OSR1, SOX1, EOMES, DDX25, and TMEM106A.

15 . The method of claim 10 , wherein the set of three or four genes comprises both of NKPD1 and KLF2.

16 . The method of claim 10 , wherein the set of three or four genes consists of MEIS1, NKPD1, ONECUT2, and KLF2.

17 . The method of claim 10 , wherein the method further comprises analyzing the bisulfite converted DNA for mutations in one or both of FGFR3 and TERT.

18 . The method of claim 10 , wherein the set of one or more reference genes comprises one or more of CTNS, TOP3A, COL2A and SLC24A3.

19 . The method of claim 10 , wherein the set of three or four genes consists of MEIS1, NKPD1, and KLF2.

Assignments (3)
TERMINATION AND RELEASE OF SECURITY INTEREST IN PATENT RIGHTS (REEL/FRAME 69898/0380) Recorded Mar 27, 2026
From: JPMORGAN CHASE BANK, N.A.
To: GENOMIC HEALTH, INC.
Reel/Frame 075294/0821 →
PATENT SECURITY AGREEMENT Recorded Jan 14, 2025
From: GENOMIC HEALTH, INC.
To: JPMORGAN CHASE BANK, N.A.
Reel/Frame 069898/0380 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 9, 2023
From: LOPATIN, MARGARITA; TSIATIS, ATHANASIOS; SILK, CHRISTOPHER N.; MILLER, DAVID P.; CRAGER, MICHAEL; FEBBO, PHILLIP; KNEZEVIC, DEJAN
To: GENOMIC HEALTH, INC.
Reel/Frame 064538/0517 →
Continuity (3)
Continuation 16612926
Provisional Application 62508274 · May 18, 2017
Related Publication 20230374604A1 · Nov 23, 2023
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