IP Library Granted Patent US 12,280,107
Granted Patent B2
US 12,280,107 · App. 18/169,632 · Granted Apr 22, 2025

Pneumococcal conjugate vaccine formulations

Inventors: William J. Smith (Harleysville, PA); Cecilia Giovarelli (Allentown, PA); Denise K. Nawrocki (Annandale, NJ)
Assignee: Merck Sharp & Dohme LLC
A61K39/385A61K47/10A61K47/20A61K47/26A61K47/36C07K1/1072C07K14/3156A61K2039/55A61K2039/6037A61K2039/70
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 12,280,107
App. No.
18/169,632
Granted
Apr 22, 2025
Kind
B2
Abstract

The present invention provides pneumococcal conjugate vaccine formulations comprising surfactant systems incorporating polysorbate 20 or a combination of a poloxamer and a polyol.

Claims (18)

1. A formulation comprising:

(i) polysaccharide-protein conjugates;

(ii) a pH buffered saline solution having a pH in the range from 5.0 to 7.5;

(iii) an aluminum salt; and

(iv) 0.2% w/v polysorbate 20 (PS-20);

wherein the polysaccharide is a S. pneumoniae polysaccharide and the protein is CRM197,

wherein the conjugates are prepared by reductive amination,

wherein 24% to 100% of the conjugates (on a total protein basis) are prepared in dimethylsulfoxide (DMSO), and

wherein S. pneumoniae polysaccharide serotypes 6A, 6B and 23F are present in the formulation and are conjugated to CRM 197 and are prepared by reductive amination in DMSO.

2. A formulation comprising:

(i) polysaccharide-protein conjugates;

(ii) a pH buffered saline solution having a pH in the range from 5.0 to 7.5;

(iii) an aluminum salt; and

(iv) 0.2% w/v polysorbate 20 (PS-20);

wherein the polysaccharide is a S. pneumoniae polysaccharide and the protein is CRM197,

wherein the conjugates are prepared by reductive amination,

wherein 24% to 100% of the conjugates (on a total protein basis) are prepared in dimethylsulfoxide (DMSO), and

wherein S. pneumoniae polysaccharide serotypes 6A, 6B, 7F, 19A, 19F and 23F are present in the formulation and are conjugated to CRM197 and are prepared by reductive amination in DMSO.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 15, 2023
From: SMITH, WILLIAM J.; GIOVARELLI, CECILIA; NAWROCKI, DENISE K.
To: MERCK SHARP & DOHME CORP.
Reel/Frame 062711/0924 →
MERGER Recorded Feb 15, 2023
From: MERCK SHARP & DOHME CORP.
To: MERCK SHARP & DOHME LLC
Reel/Frame 062711/0986 →