IP Library Granted Patent US 12,472,165
Granted Patent B2
US 12,472,165 · App. 18/361,838 · Granted Nov 18, 2025

Riluzole prodrugs and their use

Inventors: Jay Edward Wrobel (Lawrenceville, NJ); Allen B. Reitz (Lansdale, PA); Jeffery Claude Pelletier (Lafayette Hill, PA); Garry Robert Smith (Royersford, PA); Haiyan Bian (Princeton, NJ)
Assignee: Biohaven Therapeutics Ltd.
A61K31/428A61K9/006A61K9/1617A61K9/2004A61K31/454A61K31/496A61K31/506A61K31/5377A61K31/541A61K38/05A61K38/06A61K40/36A61K45/06A61P25/00A61P25/28A61P35/00C07D277/82C07D417/12C07K5/06026C07K5/0806C07K5/0808C07K5/0812A61K9/0056A61K9/2018A61K9/2063A61K9/485A61K9/4858A61K9/4866A61K2300/00
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Quick Facts
Patent No.
US 12,472,165
App. No.
18/361,838
Granted
Nov 18, 2025
Kind
B2
Abstract

Pharmaceutical compositions of the invention include substituted riluzole prodrugs useful for the treatment of cancers including melanoma, breast cancer, brain cancer, and prostate cancer through the release of riluzole. Prodrugs of riluzole have enhanced stability to hepatic metabolism and are delivered into systemic circulation by oral administration, and then cleaved to release riluzole in the plasma via either an enzymatic or general biophysical release process.

Claims (10)

1 . A method for treating spinocerebellar ataxia in a subject in need of such treatment, comprising administering a riluzole prodrug to the subject, wherein said administration comprises:

releasing an effective amount of riluzole or hydrate, solvate, pharmaceutically acceptable salt, or complex thereof into blood stream of the subject; and

attenuating presynaptic glutamate release in the subject, and

wherein the prodrug is a compound that is cleaved to release riluzole in the blood stream via either an enzymatic or general biophysical release process.

2 . The method according to claim 1 , wherein the spinocerebellar ataxia is hereditary spinocerebellar ataxia.

3 . A method for treating spinocerebellar ataxia in a subject in need of such treatment, comprising administering a riluzole prodrug to the subject, wherein said administration comprises:

contacting plasma of the subject with an effective amount of riluzole or hydrate, solvate, pharmaceutically acceptable salt, or complex thereof; and

attenuating presynaptic glutamate release in the subject, and

wherein the prodrug is a compound that is cleaved to release riluzole in the plasma via either an enzymatic or general biophysical release process.

4 . The method according to claim 3 , wherein the spinocerebellar ataxia is hereditary spinocerebellar ataxia.

Assignments (1)
SECURITY INTEREST Recorded May 1, 2025
From: BIOHAVEN THERAPEUTICS LTD
To: BEETLEJUICE SA LLC, AS PURCHASER AGENT
Reel/Frame 071147/0260 →
Continuity (6)
Continuation 17367484 · Jul 5, 2021
Continuation 16689150 · Nov 20, 2019
Continuation 16449948 · Jun 24, 2019
Continuation 15549154
Provisional Application 62127684 · Mar 3, 2015
Related Publication 20230381150A1 · Nov 30, 2023
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