IP Library Granted Patent US 12,048,712
Granted Patent B2
US 12,048,712 · App. 18/381,558 · Granted Jul 30, 2024

Beta-adrenergic agonist and muscarinic antagonist compositions and methods of using

Inventors: James R. Komorowski (Trumbull, CT); Sarah Sylla (Brooklyn, NY); Devon Bernsley (New York, NY)
Assignee: Bonafide Health, LLC
A61K31/7076A61K31/235A61K36/185A61K36/31A61K36/42A61K36/54A61K38/168A61P13/06
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Quick Facts
Patent No.
US 12,048,712
App. No.
18/381,558
Granted
Jul 30, 2024
Kind
B2
Abstract

Disclosed herein are compositions for supporting bladder health and/or treating, ameliorating, preventing, or reducing overactive bladder or the symptoms associated therewith. The compositions disclosed herein comprise a beta-adrenergic receptor agonist and at least one muscarinic receptor antagonist. Also described herein are methods utilizing the aforementioned compositions.

Claims (22)

1. A composition for supporting bladder health and/or treating overactive bladder or at least one symptom associated therewith comprising an amount of a beta-adrenergic receptor agonist and an amount of at least one muscarinic receptor antagonist, wherein the beta-adrenergic receptor agonist comprises S-adenosyl-L-methionine (SAMe) and wherein the at least one muscarinic receptor antagonist is the Crataeva nurvala plant material or extract thereof and a mixture of black maca and yellow maca, wherein the mixture of black maca and yellow maca comprises a ratio of black maca to yellow maca of about 4:1 to about 1:4.

2. The composition of claim 1 , wherein the Crataeva nurvala plant material or extract thereof, the mixture of black maca and yellow maca, and the SAMe are present in a ratio of about 4:1:1 to about 4:1:4.

3. A composition for supporting bladder health and/or treating overactive bladder or at least one symptom associated therewith comprising an amount of a beta-adrenergic receptor agonist and an amount of at least one muscarinic receptor antagonist, wherein the beta-adrenergic receptor agonist comprises S-adenosyl-L-methionine (SAMe) and propyl gallate (PG), wherein SAMe and PG comprise a mixture having a ratio of SAMe to PG of about 8:1 to about 128:1, and wherein the at least one muscarinic receptor antagonist is selected from the group consisting of pumpkin seed, Crataeva nurvala plant material or an extract thereof, Lindera aggregata plant material or an extract thereof, black maca, yellow maca, phycocyanin or an extract thereof, and any combination thereof.

4. The composition of claim 3 , wherein the at least one muscarinic receptor antagonist is the Crataeva nurvala plant material or extract thereof and a mixture of black maca and yellow maca, wherein the mixture of black maca and yellow maca comprises a ratio of black maca to yellow maca of about 4:1 to about 1:4.

5. The composition of claim 4 , wherein the Crataeva nurvala plant material or extract thereof, the mixture of black maca and yellow maca, and the mixture of SAMe and PG are present in a ratio of about 4:1:1 to about 4:1:4.

6. The composition of claim 3 , wherein the at least one muscarinic receptor antagonist is Crataeva nurvala plant material or extract thereof.

7. The composition of claim 3 , wherein the at least one muscarinic receptor antagonist consists of pumpkin seed, Crataeva nurvala plant material or extract thereof, and Lindera aggregata plant material or extract thereof.

8. A dietary supplement comprising an amount of a beta-adrenergic receptor agonist and an amount of at least of one muscarinic receptor antagonist, wherein the beta-adrenergic receptor agonist comprises S-adenosyl-L-methionine (SAMe) and wherein the at least one muscarinic receptor antagonist is Crataeva nurvala plant material or extract thereof and a mixture of black maca and yellow maca, wherein the mixture of black maca and yellow maca comprises a ratio of black maca to yellow maca of about 4:1 to about 1:4.

9. The dietary supplement of claim 8 , wherein the Crataeva nurvala plant material or extract thereof, the mixture of black maca and yellow maca, and the SAMe are present in a ratio of about 4:1:1 to about 4:1:4.

10. The dietary supplement of claim 8 , wherein the dietary supplement is administered to a subject, wherein the administration of the dietary supplement treats, ameliorates, prevents, or reduces overactive bladder or at least one symptom associated therewith, wherein the at least one symptom is selected from the group consisting of urinary urgency, urinary incontinence, urge incontinence, polyuria, nocturia, bladder spasms, and any combination thereof.

11. The dietary supplement of claim 8 , wherein the dietary supplement is administered to maintain healthy levels of bladder activity and urinary frequency.

12. The dietary supplement of claim 8 , wherein the dietary supplement is administered to maintain healthy levels of one or more of urinary urgency, urinary incontinence, urge incontinence, polyuria, nocturia, bladder spasms, and any combination thereof.

13. The dietary supplement of claim 8 , wherein the dietary supplement is administered to support bladder health.

14. A dietary supplement comprising an amount of a beta-adrenergic receptor agonist and an amount of at least one muscarinic receptor antagonist, wherein the beta-adrenergic receptor agonist comprises S-adenosyl-L-methionine SAMe) and propyl gallate (PG), wherein SAMe and PG comprise a mixture having a ratio of SAMe to PG of about 8:1 to about 128:1, and wherein the at least one muscarinic receptor antagonist is selected from the group consisting of pumpkin seed, Crataeva nurvala plant material or an extract thereof, Lindera aggregata plant material or an extract thereof, black maca, yellow maca, phycocyanin or an extract thereof, and any combination thereof.

15. The dietary supplement of claim 14 , wherein the at least one muscarinic receptor antagonist is Crataeva nurvala plant material or an extract thereof and a mixture of black maca and yellow maca, wherein the mixture of black maca and yellow maca comprises a ratio of black maca to yellow maca of about 4:1 to about 1:4.

16. The dietary supplement of claim 15 , wherein the Crataeva nurvala plant material or an extract thereof, the mixture of black maca and yellow maca, and the mixture of SAMe and PG are present in a ratio of about 4:1:1 to about 4:1:4.

17. The dietary supplement of claim 14 , wherein the at least one muscarinic receptor antagonist is Crataeva nurvala plant material or extract thereof.

18. The dietary supplement of claim 14 , wherein the at least one muscarinic receptor antagonist consists of pumpkin seed, Crataeva nurvala plant material or extract thereof, and Lindera aggregata plant material or extract thereof.

19. The dietary supplement of claim 14 , wherein the dietary supplement is administered to a subject, wherein the administration of the dietary supplement treats, ameliorates, prevents, or reduces overactive bladder or at least one symptom associated therewith, wherein the at least one symptom is selected from the group consisting of urinary urgency, urinary incontinence, urge incontinence, polyuria, nocturia, bladder spasms, and any combination thereof.

20. The dietary supplement of claim 14 , wherein the dietary supplement is administered to maintain healthy levels of bladder activity and urinary frequency.

21. The dietary supplement of claim 14 , wherein the dietary supplement is administered to maintain healthy levels of one or more of urinary urgency, urinary incontinence, urge incontinence, polyuria, nocturia, bladder spasms, and any combination thereof.

22. The dietary supplement of claim 14 , wherein the dietary supplement is administered to support bladder health.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 30, 2024
From: JDS THERAPEUTICS, LLC
To: BONAFIDE HEALTH, LLC
Reel/Frame 067273/0667 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 30, 2024
From: KOMOROWSKI, JAMES R., MR.; SYLLA, SARAH; BERNSLEY, DEVON
To: JDS THERAPEUTICS, LLC
Reel/Frame 067273/0718 →
Continuity (2)
Provisional Application 63417315 · Oct 18, 2022
Related Publication 20240122958A1 · Apr 18, 2024