IP Library Patent Application 18439671
Patent Application
App. No. 18/439,671

CRYSTALLINE PHARMACEUTICAL AND METHODS OF PREPARATION AND USE THEREOF

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Quick Facts
Patent No.
US None
App. No.
18/439,671
Abstract

Novel crystalline polymorphic forms, Forms A, B, C, D, and E of a compound of Formula I, which has been found to be a potent inhibitor of LFA-1, are disclosed. Methods of preparation and uses thereof in the treatment of LFA-1 mediated diseases are also disclosed in this invention.

Claims (6)

1 - 67 . (canceled)

68 . A method for treating diabetic macular edema in a subject in need thereof, comprising administering to the subject an effective amount of a composition comprising a compound of Formula I:

or a pharmaceutically acceptable salt thereof, wherein said compound comprises a purity of greater than about 90 percent.

69 . The method of claim 68 , wherein said compound has a purity of greater than about 98 percent.

70 . The method of claim 68 , wherein said compound comprises at least about 95 percent of an S-enantiomer.

71 . The method of claim 68 , wherein said compound is a sodium salt.

Assignments (9)
ASSIGNMENT OF SECURITY INTEREST IN PATENTS PREVIOUSLY RECORDED AT REEL/FRAME (067501/0955) Recorded Aug 14, 2025
From: CITIBANK, N.A., AS RESIGNING AGENT
To: JPMORGAN CHASE BANK, N.A., AS SUCCESSOR AGENT
Reel/Frame 072460/0665 →
PATENT SECURITY AGREEMENT Recorded Jul 1, 2025
From: BAUSCH & LOMB INCORPORATED; ALDEN OPTICAL LABORATORIES, INC.; BAUSCH + LOMB IRELAND LIMITED
To: CITIBANK, N.A., AS NOTES COLLATERAL AGENT
Reel/Frame 071773/0871 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2024
From: SARCODE BIOSCIENCE, INC.
To: NOVARTIS AG
Reel/Frame 068753/0578 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2024
From: SARCODE CORPORATION
To: SARCODE BIOSCIENCE, INC.
Reel/Frame 068753/0951 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2024
From: BURNIER, JOHN; GADEK, THOMAS; NAUD, FREDERIC
To: SARCODE CORPORATION
Reel/Frame 068371/0051 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2024
From: NOVARTIS PHARMACEUTICALS CORPORATION
To: BAUSCH + LOMB IRELAND LIMITED
Reel/Frame 068754/0066 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 22, 2024
From: NOVARTIS AG
To: NOVARTIS PHARMACEUTICALS CORPORATION
Reel/Frame 068371/0982 →
INTELLECTUAL PROPERTY SECURITY AGREEMENT Recorded May 23, 2024
From: BAUSCH + LOMB IRELAND LIMITED
To: CITIBANK, N.A., AS NOTES COLLATERAL AGENT
Reel/Frame 067527/0251 →
INTELLECTUAL PROPERTY SECURITY AGREEMENT Recorded May 22, 2024
From: BAUSCH + LOMB IRELAND LIMITED
To: CITIBANK, N.A., AS COLLATERAL AGENT
Reel/Frame 067501/0955 →