IP Library Granted Patent US 12,303,557
Granted Patent B2
US 12,303,557 · App. 18/478,368 · Granted May 20, 2025

Collagenase formulations and methods of producing the same

Inventor: Karunakar Sukuru (Garnet Valley, PA)
Assignee: Endo Operations Limited
A61K38/4886A61K31/7016A61P17/00C12Y304/24003C12Y304/24007
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Quick Facts
Patent No.
US 12,303,557
App. No.
18/478,368
Granted
May 20, 2025
Kind
B2
Abstract

Disclosed herein are improved collagenase-containing formulations and methods of preparing the same. The collagenase-containing formulations comprise a collagenase, about 30 mM to about 240 mM of a disaccharide, about 50 mM to about 800 mM of mannitol, and about 6 mM to about 10 mM of a Tris-HCl. Lyophilized and reconstituted formulations are also provided.

Claims (18)

1. A formulation comprising:

a collagenase;

about 30 mM to about 240 mM of a disaccharide;

about 50 mM to about 800 mM of mannitol; and

about 6 mM to about 10 mM of Tris-HCl.

2. The formulation of claim 1 , wherein the collagenase is produced by recombinant techniques.

3. The formulation of claim 1 , wherein the disaccharide is sucrose or trehalose.

4. The formulation of claim 1 , wherein the pH of the formulation is about 7.8 to about 8.8.

5. The formulation of claim 1 , wherein the formulation comprises:

a collagenase;

about 60 mM of sucrose;

about 225 mM of mannitol; and

about 10 mM of Tris-HCl,

wherein the formulation has a pH of about 8.5.

6. The formulation of claim 1 , further comprising a surfactant selected from polysorbate 20, polysorbate 80, and poloxamer 188.

7. The formulation of claim 6 , comprising from about 0.01% to about 2% of the surfactant.

8. The formulation of claim 7 , comprising about 0.02% of the surfactant.

9. The formulation of claim 1 , wherein the formulation is liquid.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 21, 2025
From: ENDO GLOBAL AESTHETICS LIMITED
To: PALADIN PHARMA INC.
Reel/Frame 070892/0569 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 21, 2025
From: PALADIN PHARMA INC.
To: ENDO OPERATIONS LIMTED
Reel/Frame 070893/0001 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 23, 2023
From: SUKURU, KARUNAKAR
To: ENDO GLOBAL AESTHETICS LIMITED
Reel/Frame 065307/0241 →
Continuity (3)
Continuation 17419899
Provisional Application 62788916 · Jan 6, 2019
Related Publication 20240041993A1 · Feb 8, 2024
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