IP Library Granted Patent US 12,458,681
Granted Patent B2
US 12,458,681 · App. 18/731,133 · Granted Nov 4, 2025

Compositions and method for treating acute radiation syndrome

Inventor: Eytan R. Barnea (New York, NY)
Assignee: Prince Biotech, LLC
A61K38/10A61K9/0019A61K38/07A61K38/08A61K39/001C12N5/0647C12N2501/998
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Quick Facts
Patent No.
US 12,458,681
App. No.
18/731,133
Filed
May 31, 2024
Granted
Nov 4, 2025
Kind
B2
Art Unit
1654
USPC
514/7.3
Abstract

Embodiments are directed to a method of treating acute radiation syndrome comprising administering to a subject following exposure to radiation a PreImplantation factor (PIF) peptide. Some embodiments describe a method of treating acute radiation syndrome following radiation exposure comprising transplanting bone marrow that has been exposed to a PIF peptide prior to transplantation into a subject. Other embodiments describe a method of increasing engraftment of a transplanted organ, tissue, or cell by pre-exposing the organ, tissue, or cell to a PIF peptide.

Claims (44)

1 . A method of treating and/or preventing acute radiation syndrome in a subject in need thereof and that has not received a bone marrow transplant, the method comprising:

after the subject has been exposed to radiation, administering to the subject a pharmaceutical composition comprising a therapeutically effective amount of a PreImplantation Factor (PIF) peptide, and a pharmaceutically acceptable carrier, the PIF peptide being selected from the group consisting of:

SEQ ID NO:3;

SEQ ID NO:6;

SEQ ID NO:13;

SEQ ID NO:15;

SEQ ID NO:16;

SEQ ID NO:17; and

combinations thereof.

2 . A method of treating and/or preventing gastrointestinal inflammation or injury associated with acute radiation syndrome in a subject in need thereof and that has not received a bone marrow transplant, the method comprising:

after the subject has been exposed to radiation, administering to the subject a pharmaceutical composition comprising a therapeutically effective amount of a PreImplantation Factor (PIF) peptide, and a pharmaceutically acceptable carrier, the PIF peptide being selected from the group consisting of:

SEQ ID NO:3;

SEQ ID NO:6;

SEQ ID NO:13;

SEQ ID NO:15;

SEQ ID NO:16;

SEQ ID NO:17; and

combinations thereof.

3 . The method of claim 1 , wherein the therapeutically effective amount is from about 0.10 milligrams/kilograms/day to about 10.00 milligrams/kilograms/day.

4 . The method of claim 1 , wherein the therapeutically effective amount is from about 0.75 milligrams/kilograms/day to about 1.50 milligrams/kilograms/day.

5 . The method of claim 1 , wherein the therapeutically effective amount is from about 0.75 milligrams/kilograms/day to about 1.00 milligrams/kilograms/day.

6 . The method of claim 1 , wherein the pharmaceutical composition is administered within about 24 hours after the exposure to the radiation.

7 . The method of claim 1 , wherein the pharmaceutical composition is administered intermittently or continuously for a time period of from about 2 to about 14 days.

8 . The method of claim 1 , wherein the pharmaceutical composition is administered intermittently for at least about twelve weeks.

9 . The method of claim 1 , wherein the pharmaceutical composition is administered intravenously, intramuscularly, or subcutaneously.

10 . The method of claim 1 , wherein the pharmaceutical composition is administered in an intermittent or continuous infusion.

11 . The method of claim 1 , wherein the acute radiation syndrome is caused by exposure to lethal radiation.

12 . The method of claim 1 , wherein the acute radiation syndrome is caused by exposure to a radiation dose of about 100 rads to about 6000 rads.

13 . The method of claim 1 , wherein the acute radiation syndrome comprises delayed effects of acute radiation exposure, and/or damage to any organ, tissue, or cell.

14 . The method of claim 1 , wherein the acute radiation syndrome is caused by exposure to sub-lethal radiation.

15 . The method of claim 1 , wherein the PIF peptide is SEQ ID NO: 13.

16 . The method of claim 1 , wherein the therapeutically effective amount of the PIF peptide is from about 0.10 milligrams/kilograms/day to about 10.00 milligrams/kilograms/day.

17 . The method of claim 2 , wherein the pharmaceutical composition is administered intravenously, intramuscularly, or subcutaneously.

18 . A method of treating and/or preventing colon inflammation or injury associated with acute radiation syndrome in a subject in need thereof and that has not received a bone marrow transplant, the method comprising:

after the subject has been exposed to radiation, administering to the subject a pharmaceutical composition comprising a therapeutically effective amount of a PreImplantation Factor (PIF) peptide, and a pharmaceutically acceptable carrier, the PIF peptide being selected from the group consisting of:

SEQ ID NO:3;

SEQ ID NO:6;

SEQ ID NO:13;

SEQ ID NO:15;

SEQ ID NO:16;

SEQ ID NO:17; and

combinations thereof.

19 . The method of claim 17 , wherein the pharmaceutical composition is administered intravenously, intramuscularly, or subcutaneously.

20 . The method of claim 17 , wherein the therapeutically effective amount of the PIF peptide is from about 0.10 milligrams/kilograms/day to about 10.00 milligrams/kilograms/day.

Assignments (3)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 18, 2025
From: BARNEA, EYTAN R.
To: BIOINCEPT, LLC
Reel/Frame 070550/0308 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 18, 2025
From: BESKRONE, CHAPTER 7 TRUSTEE OF THE ESTATE OF BIOINCEPT, LLC, DON A.
To: PRINCE, DOUGLAS
Reel/Frame 070550/0497 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 18, 2025
From: PRINCE, DOUGLAS
To: PRINCE BIOTECH, LLC
Reel/Frame 070550/0544 →
Continuity (6)
Continuation 17472574 · Sep 10, 2021
Continuation 15512001
Provisional Application 62211660 · Aug 28, 2015
Provisional Application 62113298 · Feb 6, 2015
Provisional Application 62051077 · Sep 16, 2014
Related Publication 20240350580A1 · Oct 24, 2024
References Cited (3)
US 4629722A · Ribi · 1986 [cited by examiner]
WO WO2013106273A2 · 2013 [cited by examiner]
WO WO2015061483A2 · 2015 [cited by examiner]