IP Library Granted Patent US 12,377,091
Granted Patent B2
US 12,377,091 · App. 18/899,500 · Granted Aug 5, 2025

Compounds and combinations thereof for treating neurological and psychiatric conditions

Inventor: Herriot Tabuteau (New York, NY)
Assignee: ANTECIP BIOVENTURES II LLC
A61K31/485A61K9/0053A61K31/135A61K31/137A61K31/15A61K31/343A61K31/381
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Quick Facts
Patent No.
US 12,377,091
App. No.
18/899,500
Granted
Aug 5, 2025
Kind
B2
Abstract

Dosage forms, drug delivery systems, and methods related to sustained release of dextromethorphan or improved therapeutic effects are disclosed. Typically, bupropion or a related compound is orally administered to a human being to be treated with, or being treated with, dextromethorphan.

Claims (20)

1. A method of treating depression comprising: orally administering a dosage form daily to a human being suffering from depression; wherein the dosage form comprises dextromethorphan or a pharmaceutically acceptable salt thereof, and sertraline or a pharmaceutically acceptable salt thereof; wherein the dextromethorphan and the sertraline are the only therapeutically active agents in the dosage form; and wherein the human being is an extensive metabolizer of dextromethorphan.

2. The method of claim 1 , wherein the dosage form is orally administered for at least 8 consecutive days.

3. The method of claim 1 , wherein the depression is major depressive disorder.

4. The method of claim 1 , wherein the depression is treatment resistant depression.

5. The method of claim 1 , wherein the dosage form comprises about 25 mg to about 100 mg of the sertraline.

6. The method of claim 1 , wherein the dosage form is orally administered for at least 14 consecutive days.

7. The method of claim 1 , wherein the dosage form provides immediate release of the dextromethorphan.

8. The method of claim 1 , wherein the dosage form provides sustained release of the Desvenlafaxine.

9. The method of claim 1 , wherein the dosage form contains about 20 mg to about 50 mg of the dextromethorphan.

10. The method of claim 1 , wherein the dosage form contains about 30 mg to about 60 mg of the dextromethorphan.

11. The method of claim 1 , wherein the dosage form contains about 40 mg to about 50 mg of the dextromethorphan.

12. The method of claim 1 , wherein the dosage form contains about 50 mg to about 70 mg of the dextromethorphan.

13. The method of claim 1 , wherein the dosage form contains about 70 mg to about 100 mg of the dextromethorphan.

14. The method of claim 1 , wherein the dosage form contains about 45 mg of a dextromethorphan salt.

15. The method of claim 1 , wherein the dextromethorphan comprises a deuterium-modified dextromethorphan.

16. The method of claim 1 , wherein the dosage form is a capsule, a tablet, or a solution.

17. The method of claim 1 , wherein a dextromethorphan plasma level is increased as compared to administering the same amount of dextromethorphan alone.

18. The method of claim 1 , wherein the human being is converted to a poor metabolizer of dextromethorphan.

19. The method of claim 1 , wherein the dosage form further comprises a pharmaceutically acceptable excipient.

20. The method of claim 1 , wherein the elimination half-life of dextromethorphan increases upon orally administering the dosage form.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Nov 7, 2024
From: TABUTEAU, HERRIOT
To: ANTECIP BIOVENTURES II LLC
Reel/Frame 069326/0244 →
Cited By (6)
US 12,564,587 US 12,576,078 US 12,599,576 US 12,653,795 US 12,661,408 US 12,678,506