IP Library Granted Patent US 8,568,721
Granted Patent B2
US 8,568,721 · App. 13/462,938 · Granted Oct 29, 2013

Method of treating rheumatoid arthritis with an anti-IL-6R antibody

Inventors: Allen Radin (New York, NY); Sean Stevens (San Francisco, CA); Tammy T. Huang (Goldens Bridge, NY); Joel H. Martin (Putnam Valley, NY); Jeanette L. Fairhurst (White Plains, NY); Ashique Rafique (Yonkers, NY); Eric Smith (New York, NY); Kevin J. Pobursky (Beacon, NY); Nicholas J. Papadopoulos (LaGrangeville, NY); James P. Fandl (LaGrangeville, NY); Gang Chen (Yorktown Heights, NY); Margaret Karow (Santa Rosa Valley, CA)
Assignee: Regeneron Pharmaceuticals, Inc.
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Quick Facts
Patent No.
US 8,568,721
App. No.
13/462,938
Granted
Oct 29, 2013
Kind
B2
Abstract

The present invention provides methods of preventing or treating rheumatoid arthritis using a fully human antibody or antigen-binding fragment thereof that specifically binds human interleukin-6 receptor (hIL-6R). The methods of the present invention may include administration of a second therapeutic agent, such as one or more of a non-steroidal anti-inflammatory drug (NSAID), a glucocorticoid, a disease-modifying anti-rheumatic drug (DMARD), or a TNF-alpha antagonist, T-cell blocker, anti-CD20 antibody, an IL-1, JAK or IL-17 antagonist, or any combination thereof.

Claims (9)

1. A method for treating rheumatoid arthritis (RA) in a subject, said method comprising administering to the subject a therapeutically effective amount of a human antibody or antigen-binding fragment thereof which specifically binds to human interleukin-6 (hIL-6R), wherein the human antibody or antigen-binding fragment comprises the complementarity determining region (CDR) sequences of a heavy chain variable region (HCVR) and light chain variable region (LCVR) pair (HCVR/LCVR) set forth in SEQ ID NO:19/27.

2. The method of claim 1 , wherein the antibody or antigen-binding fragment comprises a CDR sequence combination set forth in SEQ ID NO:21/23/25/29/31/33.

3. The method of claim 1 , wherein the antibody or antigen-binding fragment comprises a HCVR/LCVR pair set forth in SEQ ID NO:19/27.

4. The method of claim 1 , wherein the human antibody or antigen-binding fragment is administered to the subject subcutaneously.

5. The method of claim 1 , further comprising administering a second therapeutic agent to the subject.

6. The method of claim 5 , wherein the antibody or antigen-binding fragment and the second therapeutic agent are administered simultaneously or sequentially.

7. The method of claim 5 , wherein the wherein the second therapeutic agent is a non-steroidal anti-inflammatory drug (NSAID), a glucocorticoid, a disease-modifying anti-rheumatic drug (DMARD), a TNF-a antagonist, a T-cell blocker, an anti-CD20 antibody, an IL-1 antagonist, or any combination thereof.

8. The method of claim 5 , wherein the second therapeutic agent is selected from the group consisting of: methotrexate; sulfasalazine; hydroxychloroquine; leflunomide; etanercept; infliximab; adalimumab; golimumab; rilonacept; anakinra; abatacept; cetiolizumab; and rituximab.

9. The method of claim 1 , wherein the therapeutically effective amount of the antibody or antigen-binding fragment is 50 mg to 200 mg.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 31, 2013
From: RADIN, ALLEN; STEVENS, SEAN; HUANG, TAMMY T.; MARTIN, JOEL H.; FAIRHURST, JEANETTE L.; RAFIQUE, ASHIQUE; SMITH, ERIC; POBURSKY, KEVIN J.; PAPADOPOULOS, NICHOLAS J.; FANDL, JAMES P.; CHEN, GANG; KAROW, MARGARET
To: REGENERON PHARMACEUTICALS, INC.
Reel/Frame 030523/0399 →
Continuity (10)
Continuation 13286261 · Nov 1, 2011
Division 12780006 · May 14, 2010
Continuation In Part 12501657 · Jul 13, 2009
Division 11809482 · Jun 1, 2007
Provisional Application 60810664 · Jun 2, 2006
Provisional Application 60843232 · Sep 8, 2006
Provisional Application 61181749 · May 28, 2009
Provisional Application 61262661 · Nov 19, 2009
Provisional Application 61297302 · Jan 22, 2010
Related Publication 20120258098A1 · Oct 11, 2012