IP Library Granted Patent US 8,003,688
Granted Patent B2
US 8,003,688 · App. 11/172,878 · Granted Aug 23, 2011

Method of treating symptoms of common cold, allergic rhinitis and infections relating to the respiratory tract

Assignee: ImmuPharm Aps
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Quick Facts
Patent No.
US 8,003,688
App. No.
11/172,878
Granted
Aug 23, 2011
Kind
B2
Abstract

The present invention relates to methods of treating conditions and/or symptoms related to common cold of the upper and/or lower respiratory tract and/or eyes. In particular the invention relates to the methods of treating conditions and/or symptoms related to common cold comprising administration of a flavonoid or administration of a flavonoid in combination with a metal. The invention furthermore describes compositions comprising a metal and a flavonoid useful for the treatment of conditions and/or symptoms relates to common cold.

Claims (17)

1. A pharmaceutical composition, effective in vivo as an antiviral agent, comprising

(1) a pharmaceutically effective amount of at least one hydroxyethylrutoside or pharmaceutically acceptable salt thereof, said hydroxyetheylrutosides or salts thereof including troxerutin or a pharmaceutically acceptable salt thereof, said amount being antivirally effective in vivo, and

(2) an amount of zinc gluconate effective in vivo to cause the in vivo antiviral effect of the composition to exceed that of the hydroxyethylrutoside(s), or salts thereof, of the composition,

wherein said composition is suitable for topical administration to the mucosal membrane of the oral cavity, and is not a solution, unless such solution is a spray.

2. The pharmaceutical composition of claim 1 which comprises a mixture of mono-, di-, tri-and tetrahydroxyethylrutosides.

3. The pharmaceutical composition of claim 1 wherein the composition is formulated as a lozenge, chewing tablet, chewing gum, spray or aerosol.

4. The composition of claim 1 , wherein the composition is formulated as a lozenge.

5. The composition of claim 1 wherein the only hydroxyethylrutoside present in the composition is troxerutin.

6. The composition of claim 1 which is a mixture of 5-10% monohydroxyethylrutoside, 30-38% dihydroxyethylrutoside, 45-55% trihydroxyethylrutoside, and 3-12% tetrahydroxyethylrutoside.

7. The composition of claim 1 wherein the hydroxyethylrutoside provides less than 10% protection of WISH cells against rhinovirus when tested in vitro according to the tetrazolium salt (MTS) method.

8. The pharmaceutical composition according to claim 1 , wherein the composition is formulated as a lozenge, chewing tablet, chewing gum, drop, spray or aerosal.

9. A method of treatment of a condition or symptoms of a condition, wherein the condition is selected from the group consisting of common cold, viral infection of the upper and/or lower respiratory tract and/or eyes, rhinitis and hay fever, said method comprising administering to an individual in need thereof a therapeutically effective amount of the composition according to claim 1 .

10. The method according to claim 9 , wherein the symptoms are one or more symptoms selected from the group consisting of cough, sneezing, muscle pain, sore throat, hoarseness, headache, malaise, chilliness, nasal discharge, nasal obstruction, pain relating to the sinuses, rhinitus, swelling of mucosal membranes and pharyngitis.

11. The method according to claim 9 , wherein the virus infection is caused by or associated with one or more viruses selected from the group consisting of adenoviruses, picornaviruses, reoviruses, orthomyxoviruses, paramyxoviruses, caliciviruses, coronaviruses, orthomyxoviruses, rhinoviruses, echovirus and coxsackie virus.

12. The method according to claim 9 , wherein the virus infection is caused by or associated with one or more viruses selected from the group consisting of coronaviruses and rhinoviruses.

13. The method according to claim 9 , wherein the virus infection is associated with a secondary bacterial infection.

14. The method according to claim 13 , wherein the bacterial infection is caused by one or more bacteria selected from the group consisting of Streptococcus pheumoniae, Streptococcus Haemolyticae, Haemophilus influenxae and Moraxella catarrhalis.

Assignments (1)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 13, 2011
From: BERG, KURT FRIMANN
To: IMMUPHARM APS
Reel/Frame 026582/0642 →
Priority Claims (5)
DK 2000 01152 · Jul 28, 2000 · national
DK 2000 01316 · Sep 4, 2000 · national
DK 2000 01935 · Dec 23, 2000 · national
DK 2001 00007 · Jan 3, 2001 · national
DK 2001 00827 · May 22, 2001 · national
Continuity (2)
Continuation 10363430
Related Publication 20050245467A1 · Nov 3, 2005