IP Library Granted Patent US 9,789,149
Granted Patent B2
US 9,789,149 · App. 11/185,246 · Granted Oct 17, 2017

Vegetation water composition for treatment of inflammatory skin conditions

Inventors: Fujio Numano (Tokyo, JP); Roberto Crea (San Mateo, CA); Tokuko S. Wiedemann (El Cerrito, CA); Catherine M. Bitler (Menlo Park, CA)
Assignee: CreAgri, Inc.
A61K36/63A61K9/2059A61K31/05
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,789,149
App. No.
11/185,246
Granted
Oct 17, 2017
Kind
B2
Abstract

Compositions obtained from vegetation water from olives and methods for treating patients suffering from an inflammatory skin disease with the compositions are described. Included are hydroxytyrosol rich compounds obtained from olive vegetation water.

Claims (14)

1. A method for treating a person suffering from an inflammatory skin condition presenting as a discrete or generalized area of skin lesions, comprising:

identifying a person suffering from such an inflammatory skin condition that has proven refractory to treatment with immunosuppressives or glucocorticoids, and

orally administering to said person, an effective amount of a pharmaceutical composition selectively enriched for hydroxytyrosol, whereby the pharmaceutical composition is produced by (i) obtaining vegetation water from olives, (ii) adding acid to the vegetation water thereby producing acidified vegetation water, (iii) incubating the acidified vegetation water for a period until the weight ratio of hydroxytyrosol to oleuropein is between 4:1 and 200:1, thereby producing incubated acidified vegetation water, and (iv) adding 90 to 360 mg of solid olive extract to the incubated acidified vegetation water thereby producing the pharmaceutical composition, wherein the pharmaceutical composition is orally administered on a daily basis over a period of at least three months so as to reduce the area of the discrete or generalized skin lesions by at least 60%.

2. The method of claim 1 , wherein the acidified vegetation water is incubated for a period until the weight ratio of hydroxytyrosol to oleuropein in the composition is between about 5:1 to 50:1.

3. The method of claim 1 , wherein said oral administration comprises orally administering said composition in tablet, capsule, or pill form.

4. The method of claim 1 , wherein said oral administration comprises orally administering said composition in liquid form.

5. The method of claim 1 , wherein the inflammatory skin condition is refractory psoriasis.

6. The method of claim 1 , wherein the inflammatory skin condition is refractory eczema.

7. The method of claim 1 , wherein the inflammatory skin condition is refractory allergic dermatitis.

8. The method of claim 1 , wherein the inflammatory skin condition is refractory photohypersensitivity dermatosis.

9. The method of claim 1 , wherein the inflammatory skin condition is refractory lichen urticatus.

10. The method of claim 1 , wherein the composition is administered at a dosage effective to deliver between about 5.4 to 10.8 mg of total polyphenols daily.

11. The method of claim 1 , wherein the composition is administered at a dosage effective to deliver between about 2.5 to 5 mg of hydroxytyrosol daily.

12. The method of claim 1 , wherein the immunosuppressive are selected from the group consisting of tacrolimus and hydroxyurea.

Assignments (7)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Sep 27, 2023
From: CARR & FERRELL LLP; VALDEVIT, EZIO
To: HIDROX, LLC
Reel/Frame 065045/0622 →
SECURITY INTEREST Recorded Mar 1, 2023
From: 2199933 ONTARIO INC.
To: CARR AND FERRELL LLP; VALDEVIT, EZIO
Reel/Frame 062837/0081 →
SECURITY INTEREST Recorded Sep 26, 2022
From: OLIPHENOL, LLC
To: RIMON, P.C.
Reel/Frame 061541/0012 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 28, 2019
From: CALISCANA, LLC
To: OLIPHENOL, LLC
Reel/Frame 048464/0225 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2019
From: CREAGRI, INC.
To: CREA, ROBERTO
Reel/Frame 048460/0378 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 27, 2019
From: CREA, ROBERTO
To: CALISCANA, LLC
Reel/Frame 048460/0767 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 6, 2006
From: NUMANO, FUJIO; CREA, ROBERTO; WIEDEMANN, TOKUKO S.; BITLER, CATHERINE M.
To: CREAGRI, INC.
Reel/Frame 017638/0096 →
Continuity (1)
Related Publication 20070020350A1 · Jan 25, 2007