IP Library Granted Patent US 7,981,414
Granted Patent B2
US 7,981,414 · App. 11/659,009 · Granted Jul 19, 2011

Anti-inflammatory dAb

Assignee: Cephalon Australia Pty Ltd
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Quick Facts
Patent No.
US 7,981,414
App. No.
11/659,009
Granted
Jul 19, 2011
Kind
B2
Abstract

The present invention provides a recombinant domain antibody (dAb) which binds to human TNF-α, the dAb comprising an immunoglobulin heavy or light chain variable domain, wherein the variable domain comprises at least one complementarity determining region (CDR) having a sequence derived from a New World primate.

Claims (59)

1. A recombinant domain antibody (dAb) which binds to human TNF-α, wherein the dAb has a sequence selected from the group consisting of:

(SEQ ID No: 8)

DIQMTQSPSSLSASVGDRVTITCRASQAIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR;

(SEQ ID No: 9)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLLPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR;

(SEQ ID No: 10)

DIQMTQSPSSLSASVGDRVTITCRASQAIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLLPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR;

(SEQ ID No: 50)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKPPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR;

(SEQ ID No: 51)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGRGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR;

and

(SEQ ID No: 52)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLVPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

2. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 10)

DIQMTQSPSSLSASVGDRVTITCRASQAIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLLPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

3. A pharmaceutical composition comprising an effective amount of a recombinant domain antibody (dAb) according to claim 1 , together with a pharmaceutically acceptable carrier or diluent.

4. A method for detecting human TNF-α in a sample comprising contacting the sample with an effective amount of a recombinant dAb according to claim 1 and detecting the amount of bound dAb.

5. The method according to claim 4 wherein the sample is a biological sample.

6. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 8)

DIQMTQSPSSLSASVGDRVTITCRASQAIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

7. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 9)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLLPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

8. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 50)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKPPKLLIYS

ASNLETGVPSRFSGSGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

9. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 51)

DIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIYS

ASNLETGVPSRFSGRGSGTDFTLTISSLQPEDFATYYCQQVVWRPFTFGQ

GTKVEIKR.

10. A recombinant dAb according to claim 1 wherein the dAb has the sequence:

(SEQ ID No: 52)

ADIQMTQSPSSLSASVGDRVTITCRASQSIDSYLHWYQQKPGKAPKLLIY

SASNLETGVPSRFSGSGSGTDFTLTISSLVPEDFATYYCQQVVWRPFTFG

QGTKVEIKR.

Assignments (6)
CHANGE OF NAME Recorded Jul 7, 2010
From: ARANA THERAPEUTICS PTY LTD
To: CEPHALON AUSTRALIA PTY LTD
Reel/Frame 024647/0286 →
CHANGE OF NAME Recorded Jul 7, 2010
From: ARANA THERAPEUTICS LIMITED
To: ARANA THERAPEUTICS PTY LTD
Reel/Frame 024647/0289 →
CHANGE OF NAME Recorded Feb 4, 2008
From: PEPTECH LIMITED
To: ARANA THERAPEUTICS LIMITED
Reel/Frame 020460/0852 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 24, 2007
From: DOYLE, ANTHONY G.; JENNINGS, PHILIP A.
To: PEPTECH LIMITED
Reel/Frame 019203/0962 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 22, 2007
From: WOOLVEN, BENJAMIN P.; TOMLINSON, IAN M.; LEE, JENNIFER A.
To: DOMANTIS LIMITED
Reel/Frame 019052/0195 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 22, 2007
From: DOMANTIS LIMITED
To: PEPTECH LIMITED
Reel/Frame 019052/0266 →
Priority Claims (1)
AU 2005907124 · Dec 20, 2005 · national
Continuity (2)
Provisional Application 60817272 · Jun 28, 2006
Related Publication 20090226428A1 · Sep 10, 2009