IP Library Granted Patent US 7,514,439
Granted Patent B2
US 7,514,439 · App. 11/660,905 · Granted Apr 7, 2009

Oxime derivative and preparations thereof

Assignee: Mitsubishi Tanabe Pharma Corporation
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Quick Facts
Patent No.
US 7,514,439
App. No.
11/660,905
Granted
Apr 7, 2009
Kind
B2
Abstract

The problem of the present invention is to provide a useful compound as a glucokinase activating agent, which is the oxime derivative of the formula [I]: wherein Ring A is aryl or heteroaryl; Q is cycloalkyl, heterocycle, alkyl or alkenyl; Ring T is heteroaryl or heterocycle; R 1 and R 2 are independently hydrogen atom, halogen atom, cycloalkylsulfonyl or the like; R 3 and R 4 are independently hydrogen atom, hydroxy, oxo, halogen atom or the like; R 5 is hydrogen atom, halogen atom, cyano, nitro, tetrazolyl or the like; or a pharmaceutically acceptable salt thereof.

Claims (7)

1. A compound of the general formula:

wherein R 5A is a group of

or a pharmaceutically acceptable salt thereof.

2. A method for treating diabetes or a complication associated with diabetes, which comprises:

administering an effective dose of a compound of claim 1 or a pharmaceutically acceptable salt thereof to a patient in need thereof,

wherein said complication associated with diabetes is one or more complication selected from the group consisting of retinopathy, nephropathy, ischemic heart disease, arteriosclerosis and obesity.

3. A pharmaceutical composition comprising an effective amount of a compound of claim 1 or a pharmaceutically acceptable salt thereof as an active ingredient.

Assignments (2)
CHANGE OF NAME Recorded Nov 1, 2007
From: TANABE SEIYAKU CO., LTD.
To: MITSUBISHI TANABE PHARMA CORPORATION
Reel/Frame 020053/0662 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 23, 2007
From: SUGAWARA, KAZUTOSHI; MATSUDAIRA, TETSUJI; SUGAMA, HIROSHI; NAWANO, MASAO; OHASHI, RIKIYA
To: TANABE SEIYAKU CO., LTD.
Reel/Frame 019334/0754 →
Priority Claims (2)
JP 2005-202014 · Jul 11, 2005 · national
JP 2006-114243 · Apr 18, 2006 · national
Continuity (1)
Related Publication 20080132479A1 · Jun 5, 2008