IP Library Granted Patent US 8,586,553
Granted Patent B2
US 8,586,553 · App. 12/055,138 · Granted Nov 19, 2013

Therapies for cancer using RLIP76

Inventors: Sanjay Awasthi (Arlington, TX); Sharad S. Singhal (Arlington, TX); Sushma Yadav (Arlington, TX)
Assignee: Board of Regents, The University of Texas System
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Quick Facts
Patent No.
US 8,586,553
App. No.
12/055,138
Granted
Nov 19, 2013
Kind
B2
Abstract

The present invention is a composition identified as a region of ralA binding protein 1, wherein the region neighbors a membrane-associated portion of the ralA binding protein 1, reduces transport activity and membrane association of the ralA binding protein 1 and kills cells undergoing uncontrolled cell growth in a subject that has cells undergoing uncontrolled cell growth. The region is used to generate medicines that kill malignant cells and tumorigenic cells. Medicines may be in the form of antibodies, si-RNA and small molecules that recognize the region.

Claims (11)

1. A method of inhibiting growth of a malignant cell expressing RLIP76 comprising contacting the cell expressing RLIP76 with a composition that inhibits expression of RLIP76, wherein the composition comprises a proteoliposome, and wherein the composition comprises an anti-sense nucleic acid or double stranded siRNA molecule that targets nucleotides encoding a region of RLIP76 selected from the group consisting of SEQ ID NO:3, and SEQ ID NO:4.

2. The method of claim 1 , wherein the anti-sense nucleic acid is in a composition comprising a pharmaceutically acceptable carrier.

3. The method of claim 1 , wherein the composition comprises a liposome anti-sense nucleic acid that has the nucleic acid sequence of SEQ ID NO:5.

4. The method of claim 1 , wherein the malignant cell is a melanoma cell, a small cell lung cancer cell, a non-small cell lung cancer cell, an ovarian cancer cell, a prostate cancer cell or an adenocarcinoma cell.

5. The method of claim 1 , wherein the malignant cell is a melanoma cell.

6. The method of claim 1 , wherein the cell is in a subject.

7. The method of claim 1 , wherein the cell is in a human subject.

8. A method of inhibiting growth of a malignant cell expressing RLIP76 in a subject comprising: administering to the subject a pharmaceutically acceptable composition comprising an effective amount of an anti-sense nucleic acid that is effective to inhibit expression of RLIP76 in the malignant cell, wherein the pharmaceutically acceptable composition comprises a liposome, and wherein the anti-sense nucleic acid targets nucleotides encoding a region of RLIP76 selected from the group consisting of SEQ ID NO:4, and SEQ ID NO:3.

9. The method of claim 8 , wherein the anti-sense nucleic acid is complementary to an mRNA that encodes SEQ ID NO:22.

10. The method of claim 8 , wherein the malignant cell is a melanoma cell, a small cell lung cancer cell, a non-small cell lung cancer cell, an ovarian cancer cell, a prostate cancer cell or an adenocarcinoma cell.

11. The method of claim 8 , wherein the malignant cell is a melanoma cell.

Assignments (2)
CONFIRMATORY LICENSE Recorded Oct 17, 2012
From: THE UNIVERSITY OF TEXAS AT ARLINGTON
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 029145/0039 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 26, 2008
From: AWASTHI, SANJAY; SINGHAL, SHARAD S.; YADAY, SUSHMA
To: BOARD OF REGENTS, THE UNIVERSITY OF TEXAS SYSTEM
Reel/Frame 021167/0361 →
Continuity (7)
Continuation 11264910 · Nov 2, 2005
Continuation In Part 10714506 · Nov 13, 2003
Continuation In Part 12055138
Continuation In Part 10713578 · Nov 13, 2003
Provisional Application 60425917 · Nov 13, 2002
Provisional Application 60425814 · Nov 13, 2002
Related Publication 20100183702A1 · Jul 22, 2010