IP Library Granted Patent US 8,143,261
Granted Patent B2
US 8,143,261 · App. 12/432,224 · Granted Mar 27, 2012

Thiazolo (4,5-D) pyrimidine compounds

Assignee: AstraZeneca AB
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Quick Facts
Patent No.
US 8,143,261
App. No.
12/432,224
Granted
Mar 27, 2012
Kind
B2
Abstract

The invention provides certain thiazolopyrimidine compounds of formula (I) or a pharmaceutically acceptable salt or solvate thereof, processes and intermediates used in their preparation, pharmaceutical compositions containing them and their use in therapy.

Claims (4)

1. The compound 5-[[2,3-Difluorophenyl)methyl]thio]-7-[[(1R)-2-hydroxy-1-methylethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one, or a pharmaceutically acceptable salt thereof.

2. The sodium salt of 5-[[(2,3-Difluorophenyl)methyl]thio]-7-[[(1R)-2-hydroxy-1-methylethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one.

3. A pharmaceutical composition comprising the compound 5-[[2,3-Difluorophenyl)methyl]thio]-7-[[(1R)-2-hydroxy-1-methylethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one, or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable adjuvant, diluent, or carrier.

4. A pharmaceutical composition comprising the sodium salt of 5-[[2,3-Difluorophenyl)methyl]thio]-7-[[(1R)-2-hydroxy-1-methylethyl]amino]thiazolo[4,5-d]pyrimidin-2(3H)-one, or a pharmaceutically acceptable salt thereof, and a pharmaceutically acceptable adjuvant, diluent, or carrier.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Aug 2, 2011
From: WILLIS, PAUL ANDREW; BONNERT, ROGER VICTOR; HUNT, SIMON FRASER; WALTERS, IAIN ALISTAIR STEWART
To: ASTRAZENECA UK LIMITED
Reel/Frame 026685/0251 →
CHANGE OF NAME Recorded Aug 2, 2011
From: ASTRAZENECA UK LIMITED
To: ASTRAZENECA AB
Reel/Frame 026685/0514 →
Priority Claims (1)
SE 9903544 · Oct 1, 1999 · national
Continuity (3)
Continuation 10863995 · Jun 9, 2004
Continuation 10089571
Related Publication 20090281123A1 · Nov 12, 2009