IP Library Granted Patent US 10,300,031
Granted Patent B2
US 10,300,031 · App. 12/452,936 · Granted May 28, 2019

Pharmaceutical compositions for treating chronic pain and pain associated with neuropathy

Inventor: Chandra Ulagaraj Singh (San Antonio, TX)
Assignee: Trinity Laboratories Inc.
A61K31/195A61K31/137A61K31/485A61K31/5377
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 10,300,031
App. No.
12/452,936
Granted
May 28, 2019
Kind
B2
Abstract

The present invention provides methods and compositions for the treatment of neuropathic pain. In certain embodiments, compositions comprising an dextromethorphan (or other N-methyl-D-aspartate receptor antagonist), tramadol, and gabapentin can synergistically act to reduce pain in a human patient. Pharmaceutical compositions may also comprise a capsaicinoid, an esterified capsaicinoid, and/or a tricyclic antidepressant.

Claims (11)

1. A pharmaceutical composition comprising a synergistic combination of:

a) 35 mg of tramadol or a pharmaceutically acceptable salt thereof;

b) 35 mg of dextromethorphan or a pharmaceutically acceptable salt thereof; and

c) 90 mg of gabapentin or a pharmaceutically acceptable salt thereof.

2. The pharmaceutical composition of claim 1 , wherein the dextromethorphan, tramadol and/or gabapentin is in the form of a pharmaceutically acceptable salt.

3. The pharmaceutical composition of claim 1 , wherein the pharmaceutical composition is an oral dosage form.

4. The pharmaceutical composition of claim 3 , wherein the oral dosage form is in a form selected from the group consisting of a tablet, troche, lozenge, aqueous solution, solid or semi-solid solutions or mixture, oily suspension or solution, dispersible powder or granule, emulsion, multiparticulate formulation, syrup and elixir.

5. A method of treating diabetic neuropathy pain or fibromyalgia pain in a subject in need of such treatment comprising administering to the subject the pharmaceutical composition of claim 1 twice daily, and wherein the pharmaceutical composition is effective to treat the pain in the subject.

6. The method of claim 5 , wherein the method comprises administering the agents simultaneously.

7. The method of claim 6 , wherein the agents are administered in a single formulation.

8. The method of claim 5 , wherein the method comprises administering the agents sequentially.

Assignments (2)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 18, 2019
From: TRINITY LABORATORIES, INC.
To: LUMINUS BIOSCIENCES, INC.
Reel/Frame 048924/0728 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 28, 2010
From: SINGH, CHANDRA ULAGARAJ, DR.
To: TRINITY LABORATORIES INC.
Reel/Frame 025211/0387 →
Continuity (2)
Provisional Application 60954251 · Aug 6, 2007
Related Publication 20110039875A1 · Feb 17, 2011