IP Library Granted Patent US 9,012,410
Granted Patent B2
US 9,012,410 · App. 12/519,335 · Granted Apr 21, 2015

Method of treating intrauterine inflammation

Inventors: Yiping Han (Beachwood, OH); Hongqi Liu (Wynnewood, PA)
Assignee: Case Western Reserve University
A61K31/739A61K31/7028A61K31/7034
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 9,012,410
App. No.
12/519,335
Granted
Apr 21, 2015
Kind
B2
Abstract

A method of treating intrauterine inflammation in a subject associated with intrauterine bacterial infection includes administering to the subject a therapeutically effective amount of a toll-like receptor 4 antagonist. The therapeutically effective amount administered to the subject is an amount effective in reducing intrauterine inflammation in the subject.

Claims (10)

1. A method of inhibiting bacterial induced fetal death in a pregnant subject at risk of developing placental inflammation response associated with intrauterine bacterial infection, the method comprising:

administering to the pregnant subject with intrauterine bacterial infection a therapeutically effective amount of a toll-like receptor 4 antagonist, wherein the therapeutically effective amount is an amount effective to reduce intrauterine inflammation and inhibit bacterial induced fetal death in the pregnant subject.

2. The method of claim 1 , the toll-like receptor 4 antagonist comprising a monophosphoryl lipid A analog.

3. The method of claim 1 , the toll-like receptor 4 antagonist comprising an aminoalkyl-glucosaminide-phosphate (AGP).

4. The method of claim 3 , the AGP comprising the structure:

or a pharmaceutically acceptable salt or phosphate ester thereof.

5. The method of claim 1 wherein the toll-like receptor 4 antagonist is administered to the subject by intravenous infusion.

6. The method of claim 1 , wherein the toll-like receptor 4 antagonist is administered to the subject topically.

7. The method of claim 1 , wherein the bacterial induced fetal death comprising gram negative bacterial induced fetal death.

8. The method of claim 7 , wherein the gram negative bacteria is fusobacterium nucleatum.

Assignments (1)
CONFIRMATORY LICENSE Recorded Feb 24, 2014
From: CASE WESTERN RESERVE UNIVERSITY
To: NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT
Reel/Frame 032279/0047 →
Continuity (2)
Provisional Application 60874758 · Dec 13, 2006
Related Publication 20100035829A1 · Feb 11, 2010