IP Library Granted Patent US 8,389,525
Granted Patent B2
US 8,389,525 · App. 12/774,230 · Granted Mar 5, 2013

Small molecules for inhibition of protein kinases

Inventors: Renee Desai (Easton, PA); Ketan Desai (Easton, PA)
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Quick Facts
Patent No.
US 8,389,525
App. No.
12/774,230
Granted
Mar 5, 2013
Kind
B2
Abstract

The invention provides compounds that inhibit protein kinases, prodrugs of the compounds, intermediates and methods of synthesizing the compounds and/or prodrugs, pharmaceutical compositions including the compounds and/or prodrugs and methods of using the compounds and/or prodrugs in a variety of contexts, including, for example, in the treatment and/or prevention of various diseases that are responsive to protein kinase inhibition and/or that are mediated, at least in part, by inappropriate kinase activity.

Claims (4)

1. A pharmaceutical composition comprising the compound

polymorphs thereof, salts thereof, hydrates thereof, and solvates thereof and at least one of a pharmaceutically acceptable carrier, a diluent and an excipient, wherein the composition is in the form of lozenges, tablets, films or capsules.

2. A method of inhibiting a Syk kinase in an animal, comprising the step of administering to the animal an amount of a composition of claim 1 effective to inhibit a Syk kinase.

3. The method of claim 2 , wherein the animal is a human.

Assignments (3)
CHANGE OF NAME Recorded Feb 12, 2015
From: VOLTARRA PHARMACEUTICALS, INC.
To: LEVOLTA PHARMACEUTICALS, INC.
Reel/Frame 034983/0032 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 13, 2014
From: IMC BIOTECHNOLOGY, INC.
To: VOLTARRA PHARMACEUTICALS, INC.
Reel/Frame 031949/0209 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 13, 2014
From: DESAI, KETAN; DESAI, RENEE
To: IMC BIOTECHNOLOGY, INC.
Reel/Frame 031980/0228 →
Continuity (1)
Related Publication 20110275645A1 · Nov 10, 2011