IP Library Granted Patent US 8,551,949
Granted Patent B2
US 8,551,949 · App. 12/844,721 · Granted Oct 8, 2013

Methods for treatment of pain

Inventors: Lawrence R. Toll (Redwood City, CA); David C. Yeomans (Sunnyvale, CA); Martin S. Angst (Palo Alto, CA); Daniel I. Jacobs (Mountain View, CA)
Assignee: Nocicepta LLC
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Quick Facts
Patent No.
US 8,551,949
App. No.
12/844,721
Granted
Oct 8, 2013
Kind
B2
Abstract

The invention provides for methods and compositions for treatment of pain via craniofacial mucosal administration of an analgesic compound (e.g. a non-opioid analgesic peptide, an NOP agonist or N/OFQ). Intranasal administration of certain analgesic peptides such as N/OFQ results in global analgesic effects.

Claims (18)

1. A method for the treatment of pain comprising administering to an individual in need thereof an effective dose of N/OFQ via intranasal administration, provided when the pain is a trigeminal nerve-associated pain, the N/OFQ is not co-administered with an oxytocin peptide.

2. The method of claim 1 , wherein said treatment comprises treatment of a trigeminal pain, a somatic pain, a neuropathic pain or a visceral pain.

3. The method of claim 2 , wherein said treatment comprises treatment of a trigeminal pain.

4. The method of claim 2 , wherein said treatment comprises treatment of a somatic pain.

5. The method of claim 2 , wherein said treatment comprises treatment of a neuropathic pain.

6. The method of claim 2 , wherein said treatment comprises treatment of a visceral pain.

7. The method of claim 1 , wherein said treatment comprises treatment of an acute pain or a chronic pain.

8. The method of claim 7 , wherein said treatment comprises treatment of an acute pain.

9. The method of claim 7 , wherein said treatment comprises treatment of a chronic pain.

10. The method of claim 1 , wherein the pain is a craniofacial pain or a head pain.

11. The method of claim 10 , wherein the craniofacial pain or the head pain is caused by temporomandibular joint disorder (TMJ), migraine or trigeminal neuralgia.

12. The method of claim 11 , wherein the craniofacial pain or the head pain is caused by temporomandibular joint disorder (TMJ).

13. The method of claim 11 , wherein the craniofacial pain or the head pain is caused by migraine.

14. The method of claim 11 , wherein the craniofacial pain or the head pain is caused by trigeminal neuralgia.

15. The method of claim 1 , wherein N/OFQ is administered as a pharmaceutical composition.

16. The method of claim 15 , wherein the pharmaceutical composition further comprises one or more pharmaceutically acceptable excipients, adjuvants, diluents or stabilizers.

17. The method of claim 15 , wherein the pharmaceutical composition further comprises at least one protease inhibitor and/or at least one absorption enhancer.

18. The method of claim 1 , wherein the administration results in reduction of a pain rating on the VAS of 30% or more.

Assignments (5)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jul 26, 2024
From: TONIX PHARMACEUTICALS HOLDING CORP.
To: TONIX PHARMA LIMITED
Reel/Frame 068094/0984 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jun 24, 2020
From: NOCICEPTA LLC
To: TONIX PHARMACEUTICALS HOLDING CORP.
Reel/Frame 053030/0087 →
CHANGE OF NAME Recorded May 15, 2013
From: NOCICEPTIN LLC
To: NOCICEPTA LLC
Reel/Frame 030426/0815 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 15, 2013
From: TRIGEMINA, INC.
To: NOCICEPTIN LLC
Reel/Frame 030426/0818 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Oct 7, 2010
From: TOLL, LAWRENCE R.; YEOMANS, DAVID C.; ANGST, MARTIN S.; JACOBS, DANIEL I.
To: TRIGEMINA, INC.
Reel/Frame 025110/0437 →
Continuity (2)
Provisional Application 61228946 · Jul 27, 2009
Related Publication 20110021426A1 · Jan 27, 2011