IP Library Granted Patent US 8,716,483
Granted Patent B2
US 8,716,483 · App. 12/918,099 · Granted May 6, 2014

Compounds that are ERK inhibitors

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Quick Facts
Patent No.
US 8,716,483
App. No.
12/918,099
Granted
May 6, 2014
Kind
B2
Abstract

Disclosed are the ERK inhibitors of formula 1.0: and the pharmaceutically acceptable salts, and solvates thereof. Q is a tetrahydropyridinyl ring. All other substitutents are as defined herein. Also disclosed are methods of treating cancer using the compounds of formula 1.0.

Claims (16)

1. A compound of the formula:

or a pharmaceutically acceptable salt thereof.

2. The compound of claim 1 wherein said compound is:

3. A compound of the formula:

or a pharmaceutically acceptable salt thereof.

4. The compound of claim 3 wherein said compound is:

5. A compound of the formula:

or a pharmaceutically acceptable salt thereof.

6. The compound of claim 5 wherein said compound is:

7. A pharmaceutical composition comprising the compound of claim 1 .

8. A pharmaceutical composition comprising the compound of claim 3 .

9. A pharmaceutical composition comprising the compound of claim 5 .

10. A compound of the formula:

or a pharmaceutically acceptable salt thereof.

11. The compound of claim 10 wherein the compound is:

12. A pharmaceutical composition comprising the compound of claim 10 .

Assignments (3)
MERGER Recorded Aug 8, 2022
From: MERCK SHARP & DOHME CORP.
To: MERCK SHARP & DOHME LLC
Reel/Frame 061102/0145 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 17, 2014
From: SAMATAR, AHMED A
To: SCHERING CORPORATION
Reel/Frame 032450/0375 →
CHANGE OF NAME Recorded Aug 30, 2012
From: SCHERING CORPORATION
To: MERCK SHARP & DOHME CORP.
Reel/Frame 028884/0151 →