IP Library Granted Patent US 8,414,869
Granted Patent B2
US 8,414,869 · App. 12/957,016 · Granted Apr 9, 2013

Melanin promoting topical composition

Inventor: Nicholas V. Perricone (Meriden, CT)
Assignee: N.V. Perricone LLC
View Patent ↗
Loading inventors, assignments & file history…
Monitor This Case
Get email alerts when status or documents change.
Order Certified Copies
Most orders are placed with the USPTO same day — all within 24 business hours.
Order via The Patent Place →
Pre-filled with this patent's details
Quick Facts
Patent No.
US 8,414,869
App. No.
12/957,016
Granted
Apr 9, 2013
Kind
B2
Abstract

The invention provides sunless tanning compositions for application to skin comprising an effective amount of at least one dopamine precursor, an effective amount of curcumin and a dermatologically acceptable carrier. Methods for preparation of said compositions are disclosed. When applied to the skin, the compositions may be used darken skin.

Claims (27)

1. A sunless tanning composition for application to skin comprising: a melanin modulator that consists essentially of an effective amount of at least one dopamine precursor selected from tyrosine, N-Acetyl tyrosine and phenylalanine, and an effective amount of curcumin and a water-based dermatologically acceptable carrier.

2. The composition of claim 1 , wherein the dopamine precursor is present from about 1 to about 30 percent by weight of the tanning composition.

3. The composition of claim 2 , wherein the dopamine precursor is present from about 5 to about 20 percent by weight of the tanning composition.

4. The composition of claim 3 , wherein the dopamine precursor is present from about 10 to about 15 percent by weight of the tanning composition.

5. The cosmetic composition of claim 1 , wherein the dopamine precursor is N-Acetyl tyrosine.

6. The composition of claim 1 , wherein the dopamine precursor is a combination of N-Acetyl tyrosine and phenylalanine.

7. The composition of claim 1 , wherein the curcumin is present from about 0.05 to about 10 percent by weight of the tanning composition.

8. The composition of claim 7 , wherein the curcumin is present from about 1.0 to about 5 percent by weight of the tanning composition.

9. The composition of claim 8 , wherein curcumin is present at about 2.0 percent by weight of the tanning composition.

10. The composition of claim 1 , further comprising phenylisothiocyanate.

11. The composition of claim 10 , wherein the phenylisothiocyanate is present from about 0.5 to about 10.0 percent by weight of the tanning composition.

12. The composition of claim 11 , wherein the phenylisothiocyanate is present from about 1.0 to about 8.0 percent by weight of the tanning composition.

13. The composition of claim 12 , wherein the phenylisothiocyanate is present from about 2.0 to about 5.0 percent by weight of the tanning composition.

14. The composition of claim 1 , wherein the dermatologically acceptable carrier comprises one or more agents selected from the group consisting of: sodium hyaluronate, phosphatidylcholine, isopropyl palmitate, cetearyl alcohol, glycerol monostearate, shae butter, squalane, silicone and dimethyl ethanolamine.

15. The composition of claim 1 further comprising one or more agents selected from the group consisting of: α-hydroxy acids, caffeine, vitamin D3, quercertin, sulforaphanes, and a blend of magnesium aspartate and zinc gluconate and copper gluconate.

16. The composition of claim 1 , wherein the pH of the composition is in the range from about 2.5 to about 6.0.

17. The composition of claim 16 , wherein the pH of the composition is in the range from about 3.0 to about 5.5.

18. The composition of claim 17 , wherein the pH of the composition is in the range from about 3.8 to about 5.0.

19. The composition of claim 1 , wherein the composition is a lotion.

20. A sunless tanning composition comprising:

about 10 to about 15 percent by weight dopamine precursor;

about 1 to about 3 percent by weight curcumin; and

about 4 to about 6 percent by weight phenylisothiocyanate;

the balance being essentially water, wherein said dopamine precursor is selected from the group consisting of tyrosine, N-Acetyl tyrosine, phenylalanine, and mixtures thereof.

21. A method for preparing a water-based sunless tanning composition comprising a water phase, an oil phase, an aqueous DMAE mixture, an effective amount of a dopamine precursor selected from tyrosine, N-Acetyl tyrosine and phenylalanine, an effective amount of curcumin, and preservatives, comprising the steps of: adding the water phase to the oil phase; mixing the water phase with the oil phase; cooling to 38-40° C.; adding the DMAE mixture at temperature of about 38° C.; adding the dopamine precursors and curcumin to the resulting mixture at a temperature of about 35° C.; homogenizing; adding preservatives; and q.s. to 100.00 with water.

22. A method of darkening skin, the method comprising the step of administering to the skin a water-based composition comprising an effective amount of at least one dopamine precursor selected from tyrosine, N-Acetyl tyrosine and phenylalanine and an effective amount of curcumin acting in synergy with said dopamine precursor to upregulate melanin production.

23. The method of claim 22 , wherein the dopamine precursor is present from about 10 to about 15 percent by weight and the curcumin is present from about 1.0 to about 5 percent by weight.

Assignments (5)
RELEASE OF SECURITY INTEREST Recorded Nov 20, 2024
From: THE NORTHWESTERN MUTUAL LIFE INSURANCE COMPANY
To: N.V. PERRICONE LLC
Reel/Frame 069335/0366 →
RELEASE OF SECURITY INTEREST Recorded Jun 5, 2015
From: MUFG UNION BANK, N.A., AS AGENT FORMERLY KNOWN AS UNION BANK, N.A., AS AGENT
To: N.V. PERRICONE LLC
Reel/Frame 035794/0978 →
SECURITY INTEREST Recorded Jun 5, 2015
From: N.V. PERRICONE LLC
To: THE NORTHWESTERN MUTUAL LIFE INSURANCE COMPANY, AS ADMINISTRATIVE AGENT
Reel/Frame 035833/0948 →
SECURITY INTEREST Recorded Jun 2, 2014
From: N.V. PERRICONE LLC
To: UNION BANK, N.A., AS ADMINISTRATIVE AGENT FOR THE LENDERS
Reel/Frame 033075/0393 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Mar 22, 2011
From: PERRICONE, NICHOLAS V.
To: N.V. PERRICONE LLC
Reel/Frame 026001/0275 →
Continuity (1)
Related Publication 20120134938A1 · May 31, 2012