IP Library Granted Patent US 9,290,461
Granted Patent B2
US 9,290,461 · App. 12/997,004 · Granted Mar 22, 2016

Crystalline modifications of prothioconazole

Inventors: Sharona Zamir (Omer, IL); Doron Mason (Othniel, IL); Inna Faktorovitch (Beer Sheva, IL)
Assignee: ADAMA MAKHTESHIM LTD
C07D249/12
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Quick Facts
Patent No.
US 9,290,461
App. No.
12/997,004
Granted
Mar 22, 2016
Kind
B2
Abstract

There is disclosed a crystalline DMSO solvate of prothioconazole as well as amorphous prothioconazole. Methods for making these solid forms, microbicidal compositions comprising them and uses thereof are also disclosed.

Claims (3)

1. A method for preparing amorphous prothioconazole, comprising heating crystalline prothioconazole until it melts, and cooling the melted prothioconazole at a rate of 3-20° C./min, to obtain amorphous prothioconazole.

2. A method according to claim 1 , wherein said cooling is effected by placing the melted prothioconazole in an environment which is at 25° C. or lower.

3. A method according to claim 1 wherein the amorphous prothioconazole obtained is characterized by a particle size diameter (d50) in the range of 20 to 200 micrometer.

Assignments (2)
CHANGE OF NAME Recorded Jan 28, 2016
From: MAKHTESHIM CHEMICAL WORKS LTD.
To: ADAMA MAKHTESHIM LTD.
Reel/Frame 037627/0451 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Jan 14, 2011
From: ZAMIR, SHARONA; MASON, DORON; FAKTOROVITCH, INNA
To: MAKHTESHIM CHEMICAL WORKS LTD.
Reel/Frame 025638/0951 →
Continuity (2)
Provisional Application 61073058 · Jun 17, 2008
Related Publication 20110144172A1 · Jun 16, 2011