IP Library Granted Patent US 9,050,275
Granted Patent B2
US 9,050,275 · App. 13/009,282 · Granted Jun 9, 2015

Methods of screening for and treating autism spectrum disorders and compositions for same

Inventor: Theoharis C. Theoharides (Brookline, MA)
Assignee: Theta Biomedical Consulting & Development Co., Inc.
A61K31/00Y10T436/143333Y10T436/201666A61K31/352A61K31/451A61K31/4545A61K31/495A61K31/519A61K31/55A61K33/24A61K36/63A61K45/06G01N33/6896G01N2333/54G01N2333/70503G01N2800/28
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Quick Facts
Patent No.
US 9,050,275
App. No.
13/009,282
Granted
Jun 9, 2015
Kind
B2
Abstract

Disclosed are methods of screening for an autism spectrum disorder, compositions that inhibit the release of molecules that disrupt the blood-brain barrier, compositions for treating autism spectrum disorders, and methods of treating autism spectrum disorders.

Claims (11)

1. A method of treating an autism spectrum disorder, comprising administering to a subject in need thereof an effective amount of a composition comprising flavonoids and olive kernel extract, wherein the flavonoids are present in an amount of 10-3,000 mg per tablet or capsule and comprise luteolin, quercetin, and rutin, and optionally, a serotonin receptor antagonist, a defensin, a histamine-1 receptor antagonist, a histamine-3 receptor agonist, or an antipsychotic agent, wherein the composition inhibits brain blood vessel leakage.

2. The method of claim 1 , wherein the autism spectrum disorder is selected from the group consisting of Autism, Asperger's syndrome, atypical autism otherwise known as pervasive developmental disorder not otherwise specified (PDD-NOS), Rett syndrome, childhood disintegrative disorder, and sensory integration dysfunction.

3. The method of claim 1 , wherein the autism spectrum disorder is autism.

4. The method of claim 1 , wherein the autism spectrum disorder is Asperger's disorder.

5. The method of claim 1 , wherein the autism spectrum disorder is Rett syndrome.

6. The method of claim 1 , wherein the serotonin receptor antagonist is azatadine or cyproheptadine.

7. The method of claim 1 , wherein the histamine-1 receptor antagonist is azelastine, azatadine, hydroxyzine, merelastine, or, rupatadine.

8. The method of claim 1 , wherein the histamine-3 receptor agonist is R(−)-α-methyl histamine, N α -methyl histamine, N τ -methyl histamine, α-N α -dethylhistamine, α,β-dimethyl histamine, N α -methyl-α-(dimethyl)histamine, N α -methyl-α-(chloromethyl)histamine, or α,β-difluoro-N α -(fluoromethyl)histamine.

9. The method of claim 1 wherein the antipsychotic agent is risperidone.

10. The method of claim 1 wherein the defensin is peptide LL37.

11. The method of claim 1 , wherein the composition is administered by oral or parenteral routes.

Assignments (4)
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 12, 2022
From: THEOHARIDES, THEOHARIS C
To: THETA BIOMEDICAL CONSULTING & DEVELOPMENT CO., INC.
Reel/Frame 059570/0468 →
MERGER Recorded Apr 12, 2022
From: THETA BIOMEDICAL CONSULTING AND DEVELOPMENT CO., INC.
To: THETA BIOMEDICAL CONSULTING AND DEVELOPMENT, LLC
Reel/Frame 060005/0100 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Apr 7, 2011
From: THEOHARIDES, THEOHARIS C.
To: THETA BIOMEDICAL CONSULTING & DEVELOPMENT CO., INC.
Reel/Frame 026089/0707 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded Feb 9, 2011
From: THEOHARIDES, THEOHARIS C.
To: THETA BIOMEDICAL CONSULTING & DEVELOPMENT CO., INC.
Reel/Frame 025774/0863 →
Continuity (2)
Continuation In Part 12534571 · Aug 3, 2009
Related Publication 20110183019A1 · Jul 28, 2011