IP Library Granted Patent US 8,114,985
Granted Patent B2
US 8,114,985 · App. 13/045,685 · Granted Feb 14, 2012

Anti-MicroRNA oligonucleotide molecules

Assignee: Rockefeller University
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Quick Facts
Patent No.
US 8,114,985
App. No.
13/045,685
Granted
Feb 14, 2012
Kind
B2
Abstract

The invention relates to isolated anti-microRNA molecules. In another embodiment, the invention relates to an isolated microRNA molecule. In yet another embodiment, the invention provides a method for inhibiting microRNP activity in a cell.

Claims (20)

1. An isolated molecule comprising a maximum of fifty moieties, wherein each moiety comprises a base bonded to a backbone unit, said molecule comprising the microRNA molecule identified in SEQ ID NO: 141 or its corresponding anti-micro RNA molecule identified in SEQ ID NO: 447.

2. A molecule according to claim 1 , wherein the molecule is modified for increased nuclease resistance.

3. The molecule according to claim 1 , wherein at least one of the moieties is a modified ribonucleotide moiety.

4. The molecule according to claim 3 , wherein the modified ribonucleotide is substituted at the 2′ position.

5. The molecule according to claim 4 , wherein the substituent at the 2′ position is a C 1 to C 4 alkyl group.

6. The molecule according to claim 5 , wherein the alkyl group is methyl.

7. The molecule according to claim 5 , wherein the alkyl group is allyl.

8. The molecule according to claim 4 , wherein the substituent at the 2′ position is a C 1 to C 4 alkoxy-C 1 to C 4 alkyl group.

9. The molecule according to claim 8 , wherein the C 1 to C 4 alkoxy-C 1 to C 4 alkyl group is methoxyethyl.

10. The molecule according to claim 1 , wherein at least one of the moieties is a 2′-fluororibonucleotide moiety.

11. The molecule according to claim 3 , wherein the modified ribonucleotide has a methylene bridge between the 2′-oxygen atom and the 4′-carbon atom.

12. The molecule according to claim 1 , wherein the molecule comprises at least one modified moiety on the 5′ end.

13. The molecule according to claim 1 , wherein the molecule comprises at least two modified moieties at the 5′ end.

14. The molecule according to claim 1 , wherein the molecule comprises at least one modified moiety on the 3′ end.

15. The molecule according to claim 1 , wherein the molecule comprises at least two modified moieties at the 3′ end.

16. The molecule according to claim 1 , wherein the molecule comprises at least two modified moieties at the 5′ end and at least two modified moieties at the 3′ end.

17. The molecule according to claim 1 , wherein the molecule comprises a nucleotide cap at the 5′ end, the 3′ end or both.

18. The molecule according to claim 1 , wherein the molecule consists of the microRNA molecule identified in SEQ ID NO: 141.

19. The molecule according to claim 1 , wherein the molecule consists of the anti-micro RNA molecule identified in SEQ ID NO: 447.

20. A vector comprising an isolated nucleic acid molecule according to claim 1 .

Continuity (5)
Division 12794085 · Jun 4, 2010
Division 10589449
Continuation 10845057 · May 13, 2004
Continuation 10778908 · Feb 13, 2004
Related Publication 20110165669A1 · Jul 7, 2011