IP Library Granted Patent US 8,691,873
Granted Patent B2
US 8,691,873 · App. 13/253,503 · Granted Apr 8, 2014

Pharmaceutical formulations containing lipoic acid derivatives

Inventors: Robert G. L. Shorr (Edison, NJ); Robert J. Rodriguez (West Windsor, NJ); Rajinder Bhasin (Coram, NY)
Assignee: Cornerstone Pharmaceuticals, Inc.
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Quick Facts
Patent No.
US 8,691,873
App. No.
13/253,503
Granted
Apr 8, 2014
Kind
B2
Abstract

The invention provides a method of treating leukemia using a pharmaceutical composition containing bis-benzyl lipoate, triethanolamine, and a pharmaceutically acceptable diluent, where the bis-benzyl lipoate and triethanolamine form an ion pair.

Claims (8)

1. A method of treating leukemia, comprising administering to a patient in need thereof to treat the leukemia a therapeutically effective amount of a pharmaceutical formulation comprising:

(a) a compound of Formula I:

(b) triethanolamine; and

(c) a pharmaceutically acceptable diluent;

wherein the compound of Formula I and triethanolamine form an ion pair.

2. The method of claim 1 , wherein the diluent is selected from the group consisting of saline, a sugar solution, an alcohol, dimethylformamide, dimethylsulfoxide, dimethylacetamide, and combinations thereof.

3. The method of claim 1 , wherein the diluent is a dextrose solution.

4. The method of claim 3 , wherein the dextrose solution contains an amount of dextrose ranging from about 2.5% to about 10% by weight.

Assignments (2)
CHANGE OF NAME Recorded Aug 17, 2017
From: CORNERSTONE PHARMACEUTICALS, INC.
To: RAFAEL PHARMACEUTICALS, INC.
Reel/Frame 043582/0850 →
ASSIGNMENT OF ASSIGNOR'S INTEREST Recorded May 31, 2012
From: SHORR, ROBERT G.L.; RODRIGUEZ, ROBERT J.; BHASIN, RAJINDER
To: CORNERSTONE PHARMACEUTICALS, INC.
Reel/Frame 028295/0078 →
Continuity (3)
Continuation 12105100 · Apr 17, 2008
Provisional Application 60912605 · Apr 18, 2007
Related Publication 20120178812A1 · Jul 12, 2012